SCHEMBL1871973

SCHEMBL1871973

CC(C)(C)OC(=O)c1ccncc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.53
LMNA P02545 2/20 0.50
MAPT P10636 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA9 Q16790 1/20 0.49
CA14 Q9ULX7 1/20 0.49
ADRB2 P07550 1/20 0.47
ADRB1 P08588 1/20 0.47
ADRB3 P13945 1/20 0.47
CYP17A1 P05093 1/20 0.47
NAPRT Q6XQN6 1/20 0.46
POLB P06746 1/20 0.45
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25469660 0.84 ABCG2 (0.52) MAPTCA12CA1CA2CA9
SCHEMBL109451 0.84 CA1 (0.61) HSD17B10CYP1A2CYP2C19CA12CA1
SCHEMBL28061698 0.81 L3MBTL1 (0.54) LMNAMAPTCYP2C9CYP2C19ADRB2
Hydrazine SCHEMBL10771056 0.80 CA12 (0.62) HSD17B10LMNAMAPTCYP1A2CA12
SCHEMBL30239927 0.79 HSD17B10 (0.42) HSD17B10LMNAMAPTCYP1A2CYP2C9
SCHEMBL17541907 0.79 HSD17B10 (0.53) HSD17B10LMNAMAPTCYP1A2CYP2C9
SCHEMBL30312579 0.79 HCAR2 (0.52) CA12CA1CA2CA9CA14
SCHEMBL27659304 0.79 HCAR2 (0.52) CA12CA1CA2CA9CA14
SCHEMBL29199324 0.78 TDP1 (0.64) HSD17B10LMNAMAPTCYP1A2CYP2C19
SCHEMBL260960 0.78 TDP1 (0.64) HSD17B10LMNAMAPTCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 67 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104530088-A Tert-butyl 2-amino-6,7-dihydro-5H-thiazolo[5,4-b]pyridyl-4-carboxylate and derivatives thereof, and their synthesis method SUZHOU SHIYA BIOPHARMACEUTICALS INC 2015-04-22 CN claimed
CN-104364247-A Carboxamide compounds and their use as calpain inhibitors V ABBVIE DEUTSCHLAND 2015-02-18 CN claimed
US-5939568-A Accelerated catalysis of olefinic epoxidations THE SCRIPPS RESEARCH INSTITUTE (US) 1999-08-17 US claimed
WO-1998033786-A9 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS 1998-12-30 WO claimed
WO-1998033786-A1 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 1998-08-06 WO claimed
EP-4735431-A2 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. (US) 2026-05-06 EP disclosed
WO-2025106633-A1 TYK2 INHIBITORS BIOGEN MA INC. (US) 2025-05-22 WO disclosed
WO-2025076523-A1 RAS INHIBITORS AND METHODS OF USE THEREOF KESTREL THERAPEUTICS, INC. (US) 2025-04-10 WO disclosed
US-20250051309-A1 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. 2025-02-13 US disclosed
CN-119390658-A Preparation method and application of green synthetic light conversion material 浙江祥邦科技股份有限公司 2025-02-07 CN disclosed
CN-115850241-B Substituted heterocyclic compound containing alpha-ketone skeleton and application thereof 中国药科大学 2025-01-14 CN disclosed
WO-2025006568-A2 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. (US) 2025-01-02 WO disclosed
WO-1998033786-A9 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS 1998-12-30 WO disclosed
WO-1998033786-A1 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 1998-08-06 WO disclosed
EP-0042154-B1 NEW CEPHEM COMPOUNDS AND PROCESSES FOR PREPARATION THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-04-15 EP disclosed
US-4463000-A BACTERICIDES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1984-07-31 US disclosed
US-4457928-A BACTERICIDAL CEPHALOSPORINS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1984-07-03 US disclosed
US-4431642-A CEPHALOSPORINS; BACTERICIDES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1984-02-14 US disclosed
EP-0042154-A1 New cephem compounds and processes for preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1981-12-23 EP disclosed
US-4128651-A Bis-quaternary pyridinium-2-aldoxime salts and a process for their preparation MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1978-12-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250051309-A1 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME DUSP2, MKNK2, DUSP22 HSD17B10 2323/4885LMNA 4267/4885MAPT 3057/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.