SCHEMBL187458

SCHEMBL187458

COC(=O)/C(=C/c1ccccc1)NC(C)=O

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
LMNA P02545 2/20 0.49
ALDH1A1 P00352 4/20 0.47
TSHR P16473 1/20 0.47
AKR1C3 P42330 1/20 0.47
KDM4E B2RXH2 2/20 0.45
HPGD P15428 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
RECQL P46063 1/20 0.45
MTNR1A P48039 2/20 0.44
MTNR1B P49286 2/20 0.44
NPSR1 Q6W5P4 1/20 0.43
GLA P06280 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3682708 1.00 MEN1 (0.56) MEN1KMT2ALMNAALDH1A1TSHR
SCHEMBL186729 1.00 MEN1 (0.56) MEN1KMT2ALMNAALDH1A1TSHR
SCHEMBL8430294 0.91 MEN1 (0.47) MEN1KMT2ALMNAALDH1A1KDM4E
SCHEMBL8430296 0.91 MEN1 (0.47) MEN1KMT2ALMNAALDH1A1KDM4E
SCHEMBL16516485 0.91 MEN1 (0.49) MEN1KMT2ALMNAALDH1A1KDM4E
SCHEMBL16516487 0.91 MEN1 (0.49) MEN1KMT2ALMNAALDH1A1KDM4E
SCHEMBL16516488 0.91 MEN1 (0.49) MEN1KMT2ALMNAALDH1A1KDM4E
SCHEMBL25669721 0.88 EPHX1 (0.49) MEN1KMT2ALMNAALDH1A1KDM4E
SCHEMBL12394376 0.86 LMNA (0.49) MEN1KMT2ALMNAALDH1A1AKR1C3
SCHEMBL7522147 0.85 MEN1 (0.47) MEN1KMT2ALMNAALDH1A1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 161 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0592552-B1 CHIRAL PHOSPHOLANES VIA CHIRAL 1,4-DIOL CYCLIC SULFATES DU PONT (US) 1997-05-28 EP claimed
CN-122036790-A Chiral phosphine-acyclic phosphoramidite ligand, preparation method and application thereof 中国科学院大连化学物理研究所 2026-05-15 CN disclosed
CN-113121615-B Ferrocene boracic chiral diphosphine ligand and preparation method and application thereof 南方科技大学 2023-02-17 CN disclosed
CN-111018918-B Metal complex, intermediate, preparation method and application thereof 中国科学院上海有机化学研究所 2022-10-04 CN disclosed
US-11325875-B2 Compound having chiral spirobiindane skeleton and preparation method therefor ZHEJIANG JIUZHOU PHARM CO LTD (CN) 2022-05-10 US disclosed
EP-3865494-A1 METAL COMPLEX, INTERMEDIATE, AND PREPARATION METHOD AND APPLICATION THEREOF Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences (CN) 2021-08-18 EP disclosed
CN-113121615-A Ferrocene boracic chiral diphosphine ligand and preparation method and application thereof 南方科技大学 2021-07-16 CN disclosed
CN-111868065-A C-sterically hindered P-chirally derived organophosphorus compounds 勃艮第大学 2020-10-30 CN disclosed
CN-108339571-A P- chiral source organic phosphorus compounds 国家科学研究中心 2018-07-31 CN disclosed
CN-103797020-B P-chirality source organic phosphorus compound 国家科学研究中心 2018-01-30 CN disclosed
CN-1064047-C Chiral phosphine nitride-phosphine oxide double coordinate-bond ligand complex and the synthesis and application thereof CHENGDU ORGANIC CHEM INST (CN) 2001-04-04 CN disclosed
CN-1059211-C Chirality epoxy phosphine ligand compound and its synthesis and application CHENGDU ORGANIC CHEM INST (CN) 2000-12-06 CN disclosed
US-6037493-A Optically active diphosphines, preparation thereof according to a process for the resolution of the racemic mixture and use thereof RHONE-POULENC CHIMIE (FR) 2000-03-14 US disclosed
US-5783738-A Optically active diphosphines, preparation thereof according to a process for the resolution of the racemic mixture and use thereof RHONE-POULENC CHIMIE (FR) 1998-07-21 US disclosed
CN-1180707-A Chirality epoxy phosphine ligand compound and its synthesis and application CHENGDU ORGANIC CHEM INST (CN) 1998-05-06 CN disclosed
CN-1168888-A Chiral phosphine nitride-phosphine oxide double coordinate-bond ligand complex and the synthesis and application thereof CHENGDU ORGANIC CHEM INST (CN) 1997-12-31 CN disclosed
EP-0198397-B1 METHOD OF PRODUCING L-PHENYLALANINE KURARAY CO., LTD. (JP) 1993-01-07 EP disclosed
US-4743547-A PURITY, ENZYME HYDROLYSIS KURARAY CO., LTD. (JP) 1988-05-10 US disclosed
US-4654176-A Sulphonated chiral phosphines, their preparation and their use RHONE-POULENC SANTE (FR) 1987-03-31 US disclosed
EP-0198397-A2 Method of producing L-phenylalanine KURARAY CO., LTD. (JP) 1986-10-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11325875-B2 Compound having chiral spirobiindane skeleton and preparation method therefor REN, VKORC1, NR3C2 MEN1 1056/4885KMT2A 3799/4885LMNA 487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.