SCHEMBL18754258

SCHEMBL18754258

CC1(C)c2cc(O)c3cc(C(F)(F)F)ccc3c2-c2cc(NC(=O)c3ccccc3)cc(Br)c21

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 3/20 0.45
KCNK3 O14649 1/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MAPT P10636 4/20 0.43
LMNA P02545 3/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
MPO P05164 1/20 0.42
POLB P06746 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
XBP1 P17861 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TRPA1 O75762 1/20 0.41
CYP1A2 P05177 1/20 0.41
GAA P10253 1/20 0.41
RXFP1 Q9HBX9 3/20 0.40
PTGS1 P23219 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1962777 0.94 MAPT (0.42) P2RX1NPC1RAB9AMAPTLMNA
SCHEMBL18754293 0.88 P2RX1 (0.49) P2RX1KCNK3NPC1RAB9AMAPT
SCHEMBL1960938 0.82 MEN1 (0.44) P2RX1NPC1RAB9AMAPTLMNA
SCHEMBL29664191 0.80 MEN1 (0.32) MEN1KMT2A
SCHEMBL15807047 0.80 NQO2 (0.36) NPC1RAB9ALMNAMEN1KMT2A
SCHEMBL6113940 0.76 PTGS2 (0.31)
SCHEMBL16713281 0.75 SLC6A2 (0.44) MAPTPOLBGAA
SCHEMBL1958041 0.73 LMNA (0.33) MAPTLMNANPSR1
SCHEMBL16742523 0.72 PDK2 (0.41)
SCHEMBL2014165 0.71 AKR1C3 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651913-B1 INDENO-FUSED RING COMPOUNDS HAVING PHOTOCHROMIC PROPERTIES TRANSITIONS OPTICAL INC (US) 2017-04-19 EP disclosed