SCHEMBL18773850

SCHEMBL18773850

Cc1ccc(CN(C)C(=O)c2cccc(C)c2)cc1

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.67
MEN1 O00255 3/20 0.67
HPGD P15428 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
HSD17B2 P37059 4/20 0.53
HSD17B1 P14061 3/20 0.53
HDAC1 Q13547 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
HSP90AA1 P07900 2/20 0.51
LIMK2 P53671 2/20 0.51
LIMK1 P53667 1/20 0.51
MMP13 P45452 1/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2228587 0.91 KMT2A (0.82) KMT2AMEN1HPGDTDP1HSD17B2
SCHEMBL18773928 0.90 KMT2A (0.62) KMT2AMEN1HPGDTDP1HSD17B2
SCHEMBL18773897 0.89 KMT2A (0.69) KMT2AMEN1HPGDTDP1HSD17B2
SCHEMBL18773942 0.87 KMT2A (0.84) KMT2AMEN1HPGDHSD17B2HSP90AA1
SCHEMBL18773998 0.87 MEN1 (0.61) KMT2AMEN1HPGDTDP1HSD17B2
SCHEMBL15676751 0.87 KMT2A (0.66) KMT2AMEN1HPGDHSD17B2HSD17B1
SCHEMBL18774018 0.86 KMT2A (0.59) KMT2AMEN1HPGDTDP1HSD17B2
SCHEMBL18773985 0.84 KMT2A (0.58) KMT2AMEN1HPGDTDP1HSD17B2
SCHEMBL10268085 0.84 KMT2A (0.62) KMT2AMEN1HPGDHSD17B2HSD17B1
SCHEMBL1691687 0.83 KMT2A (0.61) KMT2AMEN1HPGDHSD17B2HSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773786-B1 FIVE-MEMBERED HETEROCYCLES USEFUL AS SERINE PROTEASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-04-26 EP disclosed