SCHEMBL18773985

SCHEMBL18773985

Cc1cccc(C(=O)N(C)Cc2ccc3ccccc3c2)c1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.58
MEN1 O00255 3/20 0.58
HSD17B2 P37059 4/20 0.51
HSD17B1 P14061 3/20 0.51
PDK1 Q15118 2/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
HPGD P15428 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
LIMK1 P53667 1/20 0.46
LIMK2 P53671 1/20 0.46
HSP90AA1 P07900 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
CDK4 P11802 1/20 0.46
CCND1 P24385 1/20 0.46
ACHE P22303 1/20 0.45
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18773897 0.86 KMT2A (0.69) KMT2AMEN1HSD17B2HSD17B1HPGD
SCHEMBL15676761 0.85 KMT2A (0.61) KMT2AMEN1HSD17B2HSD17B1PDK1
SCHEMBL2228587 0.84 KMT2A (0.82) KMT2AMEN1HSD17B2HSD17B1L3MBTL1
SCHEMBL18773850 0.84 KMT2A (0.67) KMT2AMEN1HSD17B2HSD17B1RAB9A
SCHEMBL18773900 0.84 MEN1 (0.43) KMT2AMEN1HSD17B2HSD17B1PDK1
SCHEMBL1696947 0.83 KMT2A (0.58) KMT2AMEN1HSD17B2HSD17B1PDK1
SCHEMBL1691800 0.82 KMT2A (0.57) KMT2AMEN1HSD17B2HSD17B1PDK1
SCHEMBL18970320 0.82 KMT2A (0.57) KMT2AMEN1HSD17B2HSD17B1PDK1
SCHEMBL18773942 0.81 KMT2A (0.84) KMT2AMEN1HSD17B2PDK1NPC1
SCHEMBL18773928 0.81 KMT2A (0.62) KMT2AMEN1HSD17B2HSD17B1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773786-B1 FIVE-MEMBERED HETEROCYCLES USEFUL AS SERINE PROTEASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-04-26 EP disclosed