SCHEMBL18773897

SCHEMBL18773897

Cc1cccc(CN(C)C(=O)c2cccc(C)c2)c1

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.69
MEN1 O00255 2/20 0.69
HSD17B2 P37059 7/20 0.61
HSD17B1 P14061 5/20 0.61
HSP90AA1 P07900 1/20 0.59
HPGD P15428 4/20 0.57
TDP1 Q9NUW8 1/20 0.57
LIMK1 P53667 1/20 0.52
LIMK2 P53671 1/20 0.52
ALDH1A1 P00352 2/20 0.48
POLB P06746 1/20 0.48
RECQL P46063 1/20 0.48
CDK4 P11802 1/20 0.48
CCND1 P24385 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
GAA P10253 1/20 0.48
TSHR P16473 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2228587 0.92 KMT2A (0.82) KMT2AMEN1HSD17B2HSD17B1HPGD
SCHEMBL18773963 0.90 MEN1 (0.60) KMT2AMEN1HSD17B2HSD17B1HSP90AA1
SCHEMBL18773850 0.89 KMT2A (0.67) KMT2AMEN1HSD17B2HSD17B1HSP90AA1
SCHEMBL18773985 0.86 KMT2A (0.58) KMT2AMEN1HSD17B2HSD17B1HSP90AA1
SCHEMBL18773928 0.85 KMT2A (0.62) KMT2AMEN1HSD17B2HSD17B1HPGD
SCHEMBL15645684 0.85 HSD17B2 (0.56) KMT2AMEN1HSD17B2HSD17B1HSP90AA1
SCHEMBL18773998 0.85 MEN1 (0.61) KMT2AMEN1HSD17B2HSD17B1HPGD
SCHEMBL11913144 0.83 HPGD (0.74) KMT2AMEN1HSD17B2HSD17B1HPGD
SCHEMBL18773942 0.83 KMT2A (0.84) KMT2AMEN1HSD17B2HSP90AA1HPGD
SCHEMBL18774018 0.82 KMT2A (0.59) KMT2AMEN1HSD17B2HSD17B1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773786-B1 FIVE-MEMBERED HETEROCYCLES USEFUL AS SERINE PROTEASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-04-26 EP disclosed