SCHEMBL18779659

SCHEMBL18779659

Nc1ccc(N2CCC[C@@H](N)C2)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.46
DOT1L Q8TEK3 1/20 0.45
PBK Q96KB5 1/20 0.44
HRH4 Q9H3N8 3/20 0.43
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
PIM1 P11309 2/20 0.40
PIM3 Q86V86 2/20 0.40
PIM2 Q9P1W9 2/20 0.40
ROCK2 O75116 3/20 0.40
ROCK1 Q13464 3/20 0.40
CDC42BPB Q9Y5S2 3/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
AKT1 P31749 1/20 0.40
CDC42BPA Q5VT25 1/20 0.40
PRKCQ Q04759 2/20 0.40
PRKCB P05771 1/20 0.40
PRKCA P17252 1/20 0.40
PRKCH P24723 1/20 0.40
PRKCE Q02156 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21698694 0.90 CCNC (0.45) HRH4CHRNB2CHRNA4CCNCCDK8
SCHEMBL23132877 0.86 DOT1L (0.44) MAP4K4DOT1LPBKHRH4PIM1
SCHEMBL4826795 0.83 CHRNB2 (0.55) DOT1LPBKCHRNB2CHRNA4PIM1
SCHEMBL22774088 0.83 DOT1L (0.44) MAP4K4DOT1LPBKHRH4CHRNB2
SCHEMBL4827711 0.83 CHRNB2 (0.56) MAP4K4DOT1LPBKHRH4CHRNB2
SCHEMBL25372604 0.83 DOT1L (0.44) MAP4K4DOT1LPBKHRH4CHRNB2
SCHEMBL24747237 0.83 CHRNB2 (0.40) CHRNB2CHRNA4ALOX5APFEN1
SCHEMBL25065178 0.83 MAP4K4 (0.47) MAP4K4CHRNB2CHRNA4CDK8
SCHEMBL25373756 0.83 CHRNB2 (0.56) MAP4K4DOT1LPBKHRH4CHRNB2
SCHEMBL23504190 0.83 DOT1L (0.44) MAP4K4DOT1LPBKHRH4CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9630970-B2 TYK2 inhibitors and uses thereof NIMBUS LAKSHMI, INC. (US) 2017-04-25 US disclosed