SCHEMBL187963

SCHEMBL187963

O=C(O)C1CC(F)CN1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL305909 1.00
SCHEMBL6196827 1.00
SCHEMBL901476 1.00
SCHEMBL187962 1.00
SCHEMBL900297 1.00
SCHEMBL661917 1.00
SCHEMBL16635328 1.00
SCHEMBL901466 1.00
Hydrochloric Acid SCHEMBL6201099 0.98 CYP2D6 (0.56)
Hydrochloric Acid SCHEMBL21598085 0.98 CYP2D6 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1159 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250325672-A1 ANTI-INFECTIVE BICYCLIC PEPTIDE LIGANDS BICYCLE TX LTD (GB) 2025-10-23 US claimed
US-12428447-B2 Peptide-based non-proteinaceous cargo delivery FELDAN BIO INC. (CA) 2025-09-30 US claimed
WO-2025085511-A1 SYSTEMS AND METHODS FOR POLYMER-MEDIATED ACTIVATION OF ENGINEERED CELLS UNIVERSITY OF WASHINGTON (US) 2025-04-24 WO claimed
US-20240197896-A1 SYNTHETIC PEPTIDE SHUTTLE AGENT BIOCONJUGATES FOR INTRACELLULAR CARGO DELIVERY FELDAN BIO INC. (CA) 2024-06-20 US claimed
CN-117750978-A Synthetic peptide shuttle bioconjugates for intracellular cargo delivery 费尔丹生物公司 2024-03-22 CN claimed
EP-4313159-A1 SYNTHETIC PEPTIDE SHUTTLE AGENT BIOCONJUGATES FOR INTRACELLULAR CARGO DELIVERY Feldan Bio Inc. (CA) 2024-02-07 EP claimed
US-20230399661-A1 SHUTTLE AGENT PEPTIDES OF MINIMAL LENGTH AND VARIANTS THEREOF ADAPTED FOR TRANSDUCTION OF CAS9-RNP AND OTHER NUCLEOPROTEIN CARGOS FELDAN BIO INC. (CA) 2023-12-14 US claimed
US-20230383291-A1 PEPTIDE-BASED TRANSDUCTION OF NON-ANIONIC POLYNUCLEOTIDE ANALOGS FOR GENE EXPRESSION MODULATION FELDAN BIO INC. (CA) 2023-11-30 US claimed
EP-4274839-A1 ANTI-INFECTIVE BICYCLIC PEPTIDE LIGANDS BicycleTx Limited (GB) 2023-11-15 EP claimed
CN-117062826-A Antiinfective bicyclic peptide ligands 拜斯科技术开发有限公司 2023-11-14 CN claimed
EP-1842841-A1 PROCESS FOR PRODUCTION OF FLUORO DERIVATIVE Central Glass Company, Limited (JP) 2007-10-10 EP claimed
EP-1007568-B1 COLLAGEN MIMICS WISCONSIN ALUMNI RES FOUND (US) 2007-08-29 EP claimed
WO-2007044026-A2 COMPOSITIONS COMPRISING MODIFIED COLLAGEN AND USES THEREFORE THE JOHNS HOPKINS UNIVERSITY (US) 2007-04-19 WO claimed
US-7122521-B2 COMPRISING TRIPEPTIDE UNIT OF THE FORMULA (flp-Yaa-Gly)N, WHERE Yaa IS ANY AMINO ACID, FLP IS 4(R)-FLUORO-L-PROLINE, AND N IS AT LEAST 3; INCREASED STABILITY; STRONGER TRIPLE HELIX THAN NATIVE COLLAGEN; FOR USE SUCH AS IN ARTIFICIAL SKIN WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2006-10-17 US claimed
WO-2005000872-A2 COLLAGEN MIMICS WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2005-01-06 WO claimed
US-20050004032-A1 Collagen mimics NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2005-01-06 US claimed
EP-1007568-A1 COLLAGEN MIMICS WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2000-06-14 EP claimed
US-5973112-A Collagen mimics WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 1999-10-26 US claimed
WO-1999010381-A1 COLLAGEN MIMICS WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 1999-03-04 WO claimed
US-5658885-A OLIGOPEPTIDES; ANTICOAGULANTS; ENZYME INHIBITORS; THROMBIN THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-19 US claimed