SCHEMBL661917

SCHEMBL661917

O=C(O)[C@@H]1C[C@H](F)CN1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL305909 1.00
SCHEMBL6196827 1.00
SCHEMBL901476 1.00
SCHEMBL187962 1.00
SCHEMBL900297 1.00
SCHEMBL16635328 1.00
SCHEMBL187963 1.00
SCHEMBL901466 1.00
Hydrochloric Acid SCHEMBL6201099 0.98 CYP2D6 (0.56)
Hydrochloric Acid SCHEMBL21598085 0.98 CYP2D6 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 439 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118984715-A Compositions for the treatment of macular degeneration comprising novel peptides 韩国视角生物株式会社 2024-11-19 CN claimed
EP-4450079-A1 COMPOSITION FOR TREATING MACULAR DEGENERATION COMPRISING NOVEL PEPTIDE EyebioKorea, Inc. (KR) 2024-10-23 EP claimed
US-20240298987-A1 Compounds For Molecular Imaging of Collagen Turnover and Methods Using Same YALE UNIVERSITY 2024-09-12 US claimed
US-20230303647-A1 CYCLIC CHEMERIN-9 DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2023-09-28 US claimed
CN-116396202-A Preparation method of (2S, 4S) -4-fluoropyrrolidine-2-carboxylic acid 南京优氟医药科技有限公司 2023-07-07 CN claimed
CN-116390742-A Cyclic chemokine-9 derivatives 拜耳公司 2023-07-04 CN claimed
WO-2023113300-A1 COMPOSITION FOR TREATING MACULAR DEGENERATION COMPRISING NOVEL PEPTIDE 주식회사 아이바이오코리아 2023-06-22 WO claimed
EP-4196143-A1 CYCLIC CHEMERIN-9 DERIVATIVES Bayer Aktiengesellschaft (DE) 2023-06-21 EP claimed
US-20230159622-A1 COLLAGEN MIMICS WISCONSIN ALUMNI RESEARCH FOUNDATION 2023-05-25 US claimed
WO-2022272268-A1 COMPOUNDS FOR MOLECULAR IMAGING OF COLLAGEN TURNOVER AND METHODS USING SAME YALE UNIVERSITY (US) 2022-12-29 WO claimed
EP-1007568-A1 COLLAGEN MIMICS WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2000-06-14 EP claimed
WO-1999060099-A1 AMINO ACID MODIFIED POLYPEPTIDES UNITED STATES SURGICAL CORPORATION (US) 1999-11-25 WO claimed
US-5973112-A Collagen mimics WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 1999-10-26 US claimed
US-5939458-A APPLYING AN INHIBITOR OF AMINOACYL-TRNA SYNTHETASE TO THE SKIN GILLETTE COMPANY, THE 1999-08-17 US claimed
WO-1999015136-A1 REDUCTION OF HAIR GROWTH THE GILLETTE COMPANY (US) 1999-04-01 WO claimed
WO-1999010381-A1 COLLAGEN MIMICS WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 1999-03-04 WO claimed
US-5720950-A ALKOXYLATED PROLINE ANALOG UNIVERSITY OF MEDICINE & DENTISTRY OF NEW JERSEY (US) 1998-02-24 US claimed
US-5660822-A A PROLINE ANALOG LINKED TO A POLYOXYALKYLENE ETHER THROUGH A SPACER COMPOUND SUCH AS LYSINE; CONTROLLING THE PROLIFERATION OF COLLAGEN; TIME-RELEASE AGENTS; NONTOXIC UNIVERSITY OF MEDICINE & DENTISTRY OF N.J. (US) 1997-08-26 US claimed
US-5372807-A Proline analogs administered to inhibit collagen accumulation UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 1994-12-13 US claimed
EP-0078191-B1 COLLAGEN INHIBITING COMPOSITIONS AND PROCESSES FOR MANUFACTURING AND USING THE SAME UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 1986-09-03 EP claimed