SCHEMBL18801441

SCHEMBL18801441

CC(C)c1cnc2c(c1)NC(=O)C(C)(C)C(=O)N2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 2/20 0.36
PDK2 Q15119 1/20 0.33
PDK4 Q16654 1/20 0.33
BMPR1B O00238 1/20 0.32
BMPR1A P36894 1/20 0.32
TGFBR1 P36897 1/20 0.32
ACVRL1 P37023 1/20 0.32
ACVR1 Q04771 1/20 0.32
ATAD2 Q6PL18 1/20 0.32
MARK3 P27448 1/20 0.31
FGFR1 P11362 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
XBP1 P17861 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16946150 0.78 MAP3K11 (0.38) MAP3K11PDK2PDK4ATAD2MARK3
SCHEMBL2707978 0.73 HPGD (0.37) MARK3FGFR1ALDH1A1LMNAMAPT
SCHEMBL16941382 0.72 BRD4 (0.46) MAP3K11BMPR1BTGFBR1ACVR1MARK3
SCHEMBL25093202 0.70 MAPK14 (0.40) MAP3K11
SCHEMBL2756587 0.69 PSEN1 (0.39) MEN1ALDH1A1LMNAMAPTKMT2A
SCHEMBL2707211 0.69 PSEN1 (0.41) ALDH1A1MAPTSMN1; SMN2
SCHEMBL26448707 0.69 MAPK14 (0.39) MAP3K11PDE3BPDE3A
SCHEMBL15457685 0.68 PDK2 (0.52) PDK2PDK4BMPR1BBMPR1ATGFBR1
SCHEMBL13340900 0.68 BRD4 (0.35)
SCHEMBL13072753 0.66 ATAD2 (0.42) PDK2PDK4BMPR1BBMPR1ATGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2882738-B1 NEW ANTIBACTERIAL COMPOUNDS JANSSEN SCIENCES IRELAND UC (IE) 2017-05-31 EP disclosed
EP-2882739-B1 NEW ANTIBACTERIAL COMPOUNDS JANSSEN SCIENCES IRELAND UC (IE) 2017-05-03 EP disclosed