SCHEMBL18814009

SCHEMBL18814009

NCc1ccc(C2=NN=C(c3ncccn3)NN2)cc1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.65
HRH3 Q9Y5N1 1/20 0.43
TAAR1 Q96RJ0 4/20 0.42
LOXL2 Q9Y4K0 4/20 0.42
CYP2A6 P11509 1/20 0.42
ASIC3 Q9UHC3 1/20 0.38
LTA4H P09960 1/20 0.37
AKT2 P31751 1/20 0.36
AKT1 P31749 1/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SGK1 O00141 1/20 0.34
SYK P43405 1/20 0.34
ATR Q13535 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18814004 0.84 ADRB2 (0.49) ADRB2HRH3TAAR1LOXL2CYP2A6
SCHEMBL2427481 0.79 ADRB2 (1.00) ADRB2HRH3TAAR1LOXL2CYP2A6
SCHEMBL28135249 0.77 ADRB2 (0.96) ADRB2HRH3TAAR1LOXL2CYP2A6
SCHEMBL18677320 0.77 HRH3 (0.45) ADRB2HRH3TAAR1LOXL2CYP2A6
SCHEMBL13978024 0.73 ADRB2 (0.78) ADRB2HRH3TAAR1LOXL2CYP2A6
SCHEMBL18653546 0.72 KDM4E (0.47) LOXL2KDM4ENPC1ALDH1A1TP53
SCHEMBL18814008 0.70 HRH3 (0.45) ADRB2HRH3TAAR1LOXL2CYP2A6
SCHEMBL505581 0.67 ADRB2 (0.62) ADRB2HRH3TAAR1LOXL2CYP2A6
SCHEMBL30083578 0.67 ADRB2 (0.62) ADRB2HRH3TAAR1LOXL2CYP2A6
SCHEMBL112429 0.67 ADRB2 (0.68) ADRB2TAAR1LOXL2CYP2A6SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017075055-A1 REDUCED AND OXIDIZED POLYSACCHARIDES AND METHODS OF USE THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2017-05-04 WO disclosed