SCHEMBL28135249

SCHEMBL28135249

NCc1ccc(-c2ccc(-c3ncccn3)cc2)cc1

nearest known ligand 0.96

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.96
HRH3 Q9Y5N1 1/20 0.61
TAAR1 Q96RJ0 4/20 0.58
CYP2A6 P11509 1/20 0.55
LOXL2 Q9Y4K0 5/20 0.50
CLK4 Q9HAZ1 1/20 0.45
LTA4H P09960 1/20 0.44
AOC3 Q16853 2/20 0.42
ASIC3 Q9UHC3 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ABAT P80404 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2427481 0.98 ADRB2 (1.00) ADRB2HRH3TAAR1CYP2A6LOXL2
SCHEMBL13978024 0.86 ADRB2 (0.78) ADRB2HRH3TAAR1CYP2A6LOXL2
SCHEMBL23291109 0.81 ADRB2 (0.70) ADRB2TAAR1CYP2A6LOXL2KDM4E
SCHEMBL16625771 0.81 CLK4 (0.61) ADRB2CYP2A6CLK4AOC3KDM4E
SCHEMBL29676764 0.79 ADRB2 (0.68) ADRB2TAAR1CYP2A6LOXL2CLK4
SCHEMBL112429 0.79 ADRB2 (0.68) ADRB2TAAR1CYP2A6LOXL2CLK4
SCHEMBL27278090 0.78 ADRB2 (0.67) ADRB2HRH3TAAR1CYP2A6LOXL2
SCHEMBL2274647 0.78 HRH3 (1.00) ADRB2HRH3TAAR1CYP2A6LOXL2
SCHEMBL6685962 0.78 CLK4 (0.64) ADRB2CYP2A6CLK4AOC3KDM4E
SCHEMBL16269874 0.78 ADRB2 (0.66) ADRB2HRH3TAAR1CYP2A6LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106496127-B A kind of preparation method of polysubstituted pyrimidine 苏州大学 2019-09-27 CN disclosed
CN-106496127-A A kind of preparation method of polysubstituted pyrimidine 苏州大学 2017-03-15 CN disclosed