SCHEMBL18848331

SCHEMBL18848331

CCC(C)(C)CCC(C(=O)O)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
THRB P10828 1/20 0.31
KMT2A Q03164 1/20 0.31
FFAR1 O14842 1/20 0.30
CPT2 P23786 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22059626 0.81 TSHR (0.31) ALDH1A1
SCHEMBL19772215 0.80 TSHR (0.33) ALDH1A1THRB
SCHEMBL13522614 0.79
SCHEMBL15362566 0.78 CES2 (0.34) MEN1ALDH1A1CYP1A2THRBKMT2A
SCHEMBL15362810 0.77 MEN1 (0.37) MEN1ALDH1A1CYP1A2THRBKMT2A
SCHEMBL14449317 0.76
SCHEMBL18850561 0.74 CES2 (0.41) MEN1CYP1A2KMT2A
SCHEMBL8688496 0.72 CES2 (0.48) MEN1CYP1A2KMT2A
SCHEMBL20503836 0.71 TSHR (0.42) MEN1ALDH1A1CYP1A2THRBKMT2A
SCHEMBL27644450 0.70 GGT1 (0.52) MEN1ALDH1A1CYP1A2THRBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9868758-B2 Betulinic proline imidazole derivatives as HIV inhibitors HETERO LABS LIMITED (IN) 2018-01-16 US disclosed
US-20170129917-A1 NOVEL BETULINIC PROLINE IMIDAZOLE DERIVATIVES AS HIV INHIBITORS HETERO LABS LIMITED (IN) 2017-05-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170129917-A1 NOVEL BETULINIC PROLINE IMIDAZOLE DERIVATIVES AS HIV INHIBITORS BET1, PRR12, IMPA1 MEN1 4006/4885ALDH1A1 4100/4885CYP1A2 4068/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.