SCHEMBL18861

SCHEMBL18861

COc1cccc2c1c(NS(=O)(=O)c1ccc(C)c(F)c1)nn2Cc1cccc(CNC(=O)C(C)(C)O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 20/20 1.00
CCR5 P51681 1/20 0.70
FFAR4 Q5NUL3 1/20 0.70
SLCO1B1 Q9Y6L6 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26339 0.93 CCR4 (0.86) CCR4CCR5FFAR4SLCO1B1
SCHEMBL30536 0.91 CCR4 (0.83) CCR4CCR5FFAR4SLCO1B1
SCHEMBL27059 0.89 CCR4 (1.00) CCR4CCR5FFAR4SLCO1B1
SCHEMBL12473981 0.85 CCR4 (0.75) CCR4CCR5FFAR4SLCO1B1
SCHEMBL30447 0.85 CCR4 (0.74) CCR4CCR5FFAR4SLCO1B1
SCHEMBL30230 0.83 CCR4 (0.71) CCR4CCR5FFAR4SLCO1B1
SCHEMBL30522123 0.83 CCR4 (0.98) CCR4CCR5FFAR4SLCO1B1
SCHEMBL358731 0.82 CCR4 (1.00) CCR4CCR5FFAR4SLCO1B1
SCHEMBL30241543 0.82 CCR4 (1.00) CCR4CCR5FFAR4SLCO1B1
SCHEMBL30241535 0.82 CCR4 (1.00) CCR4CCR5FFAR4SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025473-A1 CC.CHEMOKINE RECEPTOR 4 ANTAGONISTS GLAXO GROUP LIMITED (GB) 2012-03-01 WO disclosed
WO-2012025473-A1 CC.CHEMOKINE RECEPTOR 4 ANTAGONISTS GLAXO GROUP LIMITED (GB) 2012-03-01 WO disclosed