SCHEMBL18870568

SCHEMBL18870568

CC(C)(C)OC(=O)N1CC2CC1CN2c1ncc(Br)cc1C#N

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RET P07949 2/20 0.51
PIK3CD O00329 10/20 0.45
GPR119 Q8TDV5 2/20 0.44
HDAC1 Q13547 1/20 0.43
PIK3R1 P27986 2/20 0.42
PARP1 P09874 1/20 0.41
AR P10275 3/20 0.40
HSD11B1 P28845 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18838012 0.92 GPR119 (0.44) RETPIK3CDGPR119HDAC1PIK3R1
SCHEMBL30206022 0.85 GPR119 (0.47) RETPIK3CDGPR119HDAC1PARP1
SCHEMBL30206226 0.84 GPR119 (0.46) RETPIK3CDGPR119HDAC1PARP1
SCHEMBL20555810 0.84 PIK3CD (0.44) RETPIK3CDPIK3R1
SCHEMBL22772735 0.82 PIK3CD (0.54) RETPIK3CDGPR119HDAC1PIK3R1
SCHEMBL22772736 0.82 PIK3CD (0.54) RETPIK3CDGPR119HDAC1PIK3R1
SCHEMBL29353492 0.82 PIK3CD (0.54) RETPIK3CDGPR119HDAC1PIK3R1
SCHEMBL1200061 0.79 GPR119 (0.61) RETGPR119HDAC1PARP1HSD11B1
SCHEMBL1200066 0.79 GPR119 (0.61) RETGPR119HDAC1PARP1HSD11B1
SCHEMBL12740858 0.79 GPR119 (0.61) RETGPR119HDAC1PARP1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017083216-A1 CYANOPYRIDINE DERIVATIVES AS LIVER X RECEPTOR BETA AGONISTS, COMPOSITIONS, AND THEIR USE MERCK SHARP & DOHME CORP. (US) 2017-05-18 WO disclosed