SCHEMBL18872452

SCHEMBL18872452

Cc1cc(Nc2ccc(C3CCCN3C)cn2)c(=O)n(C)n1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.50
CCND1 P24385 1/20 0.50
BTK Q06187 3/20 0.43
MELK Q14680 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL611331 0.88 CDK4 (0.49) CDK4CCND1BTKMELK
SCHEMBL611330 0.88 CDK4 (0.49) CDK4CCND1BTKMELK
SCHEMBL1393129 0.80 CDK4 (0.54) CDK4CCND1BTKMELK
SCHEMBL18872599 0.78 FASN (0.45) CDK4CCND1BTK
SCHEMBL29398395 0.72 ALDH1A1 (0.52)
SCHEMBL1848739 0.72 ALDH1A1 (0.52)
SCHEMBL1848736 0.72 ALDH1A1 (0.52)
SCHEMBL12650332 0.72 HPGD (0.51) CDK4BTK
SCHEMBL5249340 0.72 CHRNA7 (0.62)
SCHEMBL29173751 0.72 CHRNA7 (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2744804-B1 INHIBITORS OF BRUTON'S TYROSINE KINASE HOFFMANN LA ROCHE (CH) 2017-05-17 EP disclosed