SCHEMBL188739

SCHEMBL188739

O=c1[nH]c(=O)c2ncn([C@@H]3O[C@H](COP(=O)(O)O)[C@@H](O)[C@H]3O)c2[nH]1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 7/20 0.66
IMPDH1 P20839 2/20 0.66
TAS1R3 Q7RTX0 3/20 0.62
TAS1R1 Q7RTX1 3/20 0.62
DNPH1 O43598 3/20 0.58
FBP1 P09467 2/20 0.58
PRKAB2 O43741 1/20 0.58
TRPM2 O94759 1/20 0.58
LDHA P00338 1/20 0.58
ADRB2 P07550 1/20 0.58
SRC P12931 1/20 0.58
ADORA1 P30542 1/20 0.58
P2RY2 P41231 1/20 0.58
P2RY1 P47900 1/20 0.58
PRKAG1 P54619 1/20 0.58
PRKAA2 P54646 1/20 0.58
PDE4D Q08499 1/20 0.58
KCNH2 Q12809 1/20 0.58
PRKAA1 Q13131 1/20 0.58
PDE3A Q14432 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL188741 1.00 IMPDH2 (0.66) IMPDH2IMPDH1TAS1R3TAS1R1DNPH1
SCHEMBL12727828 1.00 IMPDH2 (0.66) IMPDH2IMPDH1TAS1R3TAS1R1DNPH1
SCHEMBL22986473 1.00 IMPDH2 (0.66) IMPDH2IMPDH1TAS1R3TAS1R1DNPH1
SCHEMBL27862445 1.00 IMPDH2 (0.66) IMPDH2IMPDH1TAS1R3TAS1R1DNPH1
SCHEMBL4356337 1.00 IMPDH2 (0.66) IMPDH2IMPDH1TAS1R3TAS1R1DNPH1
SCHEMBL2217345 1.00 IMPDH2 (0.66) IMPDH2IMPDH1TAS1R3TAS1R1DNPH1
SCHEMBL20266268 0.99 IMPDH2 (0.65) IMPDH2IMPDH1TAS1R3TAS1R1DNPH1
SCHEMBL22635931 0.99 IMPDH2 (0.65) IMPDH2IMPDH1TAS1R3TAS1R1DNPH1
Phosphoric Acid SCHEMBL30728570 0.99 IMPDH2 (0.65) IMPDH2IMPDH1TAS1R3TAS1R1DNPH1
SCHEMBL28340155 0.99 IMPDH2 (0.65) IMPDH2IMPDH1TAS1R3TAS1R1DNPH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2194 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4223352-B1 DRUG-COATED BALLOON CATHETERS FOR BODY LUMENS UROTRONIC INC (US) 2026-05-27 EP claimed
EP-4747627-A1 METHODS AND SYSTEMS FOR PREDICTIVE CLASSIFICATION BY MASS SPECTROMETRY AND TRAINED LARGE SPECTRAL MODELS Matterworks Inc (US) 2026-05-27 EP claimed
US-20260114475-A1 ANIMAL FOOD COMPOSITIONS WITH IMPROVED PALATABILITY AND CUSTOMIZABILITY, AND METHODS FOR PREPARING THE SAME MARS, INCORPORATED (US) 2026-04-30 US claimed
US-12605342-B2 Polymer-encapsulated drug particles TONIC MEDICAL, INC. (US) 2026-04-21 US claimed
US-20250289840-A1 RNA STABILIZING SUBSTANCES AND METHODS OF USE TEAM MEDICAL, LLC 2025-09-18 US claimed
EP-4593631-A1 ANIMAL FOOD COMPOSITIONS WITH IMPROVED PALATABILITY AND CUSTOMIZABILITY, AND METHODS FOR PREPARING THE SAME Mars, Incorporated (US) 2025-08-06 EP claimed
US-12280226-B2 Drug-coated balloon catheters for body lumens UROTRONIC, INC. (US) 2025-04-22 US claimed
WO-2025072741-A1 PRESERVATIVES FOR MOLECULAR SAMPLE ANALYSIS WITH SAMPLE COLLECTION DEVICES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2025-04-03 WO claimed
CN-119733157-A Drug coated balloon catheter for non-vascular stenosis 江苏长寿棒科技有限公司 2025-04-01 CN claimed
US-20250082582-A1 POLYMER-ENCAPSULATED DRUG PARTICLES TONIC MEDICAL, INC. 2025-03-13 US claimed
US-5650403-A PURINE-BASED COMPOUNDS (TASTANDS, E.G. IOSINE, GUANOSINE AND XANTHINE-5'-PHOSPHATE) USED TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; ARTIFICIAL SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-07-22 US claimed
US-5631038-A COMPOUNDS (TASTANDS) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE ARE ADDED TO FOODS CONTAINING SODIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US claimed
EP-0661932-A4 SPECIFIC EATABLE TASTE MODIFIERS. BIORESEARCH INC (US) 1996-06-05 EP claimed
EP-0661932-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1995-07-12 EP claimed
WO-1993010677-A1 SPECIFIC EATABLE TASTE MODIFIERS BIORESEARCH, INC. (US) 1993-06-10 WO claimed
EP-0185092-B1 PROCESS FOR PREPARING 5'-GUANYLIC ACID KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-10-07 EP claimed
EP-0251489-B1 PROCESS FOR PRODUCING 5'-GUANYLIC ACID KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-07-22 EP claimed
US-5034378-A Flavor enhancers for food of sodium chloride, potassium chloride, monosodium glutamate and fibers Cox, James P. (US) 1991-07-23 US claimed
EP-0263716-A2 A process for the preparation of 5'-guanylic acid and expression vectors for use therein KYOWA HAKKO KOGYO KABUSHIKI KAISHA (JP) 1988-04-13 EP claimed
US-4577012-A ABSORPTION ON ACTIVATED CARBON, ELUTION WITH ALKALI HYDROXIDE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1986-03-18 US claimed