SCHEMBL18901170

SCHEMBL18901170

CCOC(=O)c1csc(-c2cccc(CN)c2)n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.58
GAA P10253 1/20 0.58
NPC1 O15118 5/20 0.54
CLK1 P49759 1/20 0.54
L3MBTL1 Q9Y468 2/20 0.53
MAPT P10636 3/20 0.52
POLB P06746 1/20 0.52
PKM P14618 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52
ALDH1A1 P00352 3/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
ROCK2 O75116 1/20 0.49
CYP1A2 P05177 2/20 0.47
KDM4E B2RXH2 1/20 0.46
HSP90AA1 P07900 1/20 0.46
SMN1; SMN2 Q16637 3/20 0.45
MMP1 P03956 1/20 0.44
MMP13 P45452 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27107843 0.89 RAB9A (0.67) RAB9AGAANPC1CLK1L3MBTL1
SCHEMBL27113213 0.88 RAB9A (0.58) RAB9AGAANPC1CLK1L3MBTL1
Bromide SCHEMBL27139844 0.88 RAB9A (0.66) RAB9AGAANPC1CLK1L3MBTL1
SCHEMBL12875862 0.85 RAB9A (0.59) RAB9AGAANPC1CLK1L3MBTL1
SCHEMBL2080725 0.85 RAB9A (0.68) RAB9AGAANPC1CLK1L3MBTL1
SCHEMBL14564380 0.84 RAB9A (0.58) RAB9AGAANPC1CLK1L3MBTL1
SCHEMBL2328911 0.83 L3MBTL1 (0.74) RAB9AGAANPC1CLK1L3MBTL1
SCHEMBL4726197 0.83 RAB9A (0.60) RAB9AGAANPC1CLK1L3MBTL1
SCHEMBL30807340 0.82 RAB9A (0.52) RAB9AGAANPC1CLK1L3MBTL1
SCHEMBL27109310 0.82 RAB9A (0.52) RAB9AGAANPC1CLK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3016951-B1 TRICYCLIC PYRIDO-CARBOXAMIDE DERIVATIVES AS ROCK INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-05-31 EP disclosed