SCHEMBL18901337

SCHEMBL18901337

O=C(CNI)c1sccc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPT P10636 2/20 0.44
AGTR1 P30556 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PKM P14618 1/20 0.44
KMT2A Q03164 4/20 0.41
HTT P42858 1/20 0.41
GSK3B P49841 1/20 0.40
OPRM1 P35372 1/20 0.39
ROCK2 O75116 1/20 0.38
MAPK1 P28482 1/20 0.38
ATM Q13315 1/20 0.38
CASP3 P42574 2/20 0.38
SENP8 Q96LD8 2/20 0.38
SENP7 Q9BQF6 2/20 0.38
SENP6 Q9GZR1 2/20 0.38
MEN1 O00255 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
KDR P35968 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17790208 0.82 MAPT (0.50) GAAALDH1A1MAPTAGTR1TDP1
SCHEMBL19954217 0.79 MAPT (0.44) GAAALDH1A1MAPTAGTR1TDP1
SCHEMBL17788643 0.78 MAPT (0.43) GAAALDH1A1MAPTAGTR1TDP1
SCHEMBL5868892 0.78 GAA (0.46) GAAALDH1A1MAPTAGTR1TDP1
SCHEMBL2096641 0.76 MAPT (0.46) GAAALDH1A1MAPTAGTR1TDP1
SCHEMBL10126109 0.76 MAPT (0.50) GAAALDH1A1MAPTAGTR1TDP1
SCHEMBL5034243 0.76 MAPT (0.46) GAAALDH1A1MAPTAGTR1TDP1
SCHEMBL27596936 0.74 ALDH1A1 (0.48) GAAALDH1A1MAPTAGTR1TDP1
SCHEMBL4947113 0.74 SMN1; SMN2 (0.51) GAAALDH1A1MAPTAGTR1TDP1
SCHEMBL4941117 0.74 ROCK2 (0.53) GAAALDH1A1MAPTAGTR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3016951-B1 TRICYCLIC PYRIDO-CARBOXAMIDE DERIVATIVES AS ROCK INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-05-31 EP disclosed