SCHEMBL18924386

SCHEMBL18924386

COC(=O)c1ccc(-c2ccc(C(=O)N(C)C3CCCC3)cc2)cc1F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.51
ERN1 O75460 2/20 0.46
FASN P49327 2/20 0.46
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
POLB P06746 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ACACB O00763 1/20 0.41
KCNH2 Q12809 2/20 0.40
MCHR1 Q99705 2/20 0.40
HPGD P15428 1/20 0.40
HTR2C P28335 1/20 0.40
USP30 Q70CQ3 1/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18924337 0.82 MAPK14 (0.55) MAPK14ERN1FASNALDH1A1GAA
SCHEMBL18924453 0.81 MAPK14 (0.59) MAPK14ERN1FASNALDH1A1GAA
SCHEMBL16323556 0.81 FASN (0.74) FASN
SCHEMBL19391337 0.81 FASN (0.74) FASN
SCHEMBL19391338 0.80 FASN (0.64) MAPK14ERN1FASNALDH1A1GAA
SCHEMBL18924525 0.78 KCNH2 (0.57) MAPK14ALDH1A1GAASMN1; SMN2POLB
SCHEMBL18924347 0.78 MAPK14 (0.48) MAPK14ERN1FASNALDH1A1GAA
SCHEMBL18924335 0.78 MAPK14 (0.52) MAPK14ERN1ALDH1A1GAASMN1; SMN2
SCHEMBL18924523 0.77 RXRB (0.50) MAPK14ALDH1A1GAASMN1; SMN2POLB
SCHEMBL18924563 0.76 MCHR1 (0.59) FASNALDH1A1GAASMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670142-B2 1,3-diaminocyclopentane carboxamide derivatives MERCK PATENT GMBH (DE) 2017-06-06 US disclosed