SCHEMBL18924453

SCHEMBL18924453

COC(=O)c1ccc(-c2ccc(C(=O)N(C)C3CCCC3)cc2)c(F)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.59
FASN P49327 2/20 0.46
ALDH1A1 P00352 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
GAA P10253 1/20 0.45
ERN1 O75460 1/20 0.44
POLB P06746 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
PDK2 Q15119 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
USP30 Q70CQ3 1/20 0.43
TACR1 P25103 1/20 0.41
KCNH2 Q12809 2/20 0.41
GRM2 Q14416 1/20 0.41
HPGD P15428 1/20 0.40
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18924450 0.87 MAPK14 (0.58) MAPK14FASNALDH1A1SMN1; SMN2GAA
SCHEMBL18924431 0.86 MAPK14 (0.53) MAPK14FASNALDH1A1SMN1; SMN2GAA
SCHEMBL18924386 0.81 MAPK14 (0.51) MAPK14FASNALDH1A1SMN1; SMN2GAA
SCHEMBL16323661 0.81 FASN (0.72) MAPK14FASN
SCHEMBL16365552 0.81 FASN (0.72) MAPK14FASN
SCHEMBL19391067 0.79 FASN (0.68) MAPK14FASNALDH1A1SMN1; SMN2GAA
SCHEMBL2945243 0.77 PTGS1 (0.57) ALDH1A1SMN1; SMN2ERN1NPC1RAB9A
SCHEMBL18924525 0.76 KCNH2 (0.57) MAPK14ALDH1A1SMN1; SMN2GAAPOLB
SCHEMBL18924561 0.75 MCHR1 (0.64) MAPK14ALDH1A1SMN1; SMN2GAAPOLB
SCHEMBL18924461 0.75 MAPK14 (0.47) MAPK14FASNPOLBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670142-B2 1,3-diaminocyclopentane carboxamide derivatives MERCK PATENT GMBH (DE) 2017-06-06 US disclosed