SCHEMBL18925014

SCHEMBL18925014

CC(O)c1cn(Cc2ccc(F)cc2)nn1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.45
KCNH2 Q12809 1/20 0.44
HDAC1 Q13547 1/20 0.44
PTGS2 P35354 1/20 0.44
KDM1A O60341 3/20 0.42
MAPT P10636 3/20 0.41
LMNA P02545 1/20 0.41
NOTUM Q6P988 1/20 0.41
CDC7 O00311 1/20 0.41
ROCK2 O75116 1/20 0.41
GSK3B P49841 1/20 0.41
ESRRG P62508 1/20 0.40
ALDH1A1 P00352 2/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2819525 0.86 NPC1 (0.52) HDAC1PTGS2KDM1ANOTUMESRRG
SCHEMBL18925110 0.84 CYP19A1 (0.53) SIGMAR1LMNAALDH1A1
SCHEMBL2819878 0.84 TEK (0.49) HDAC1KDM1AMAPTNOTUM
SCHEMBL18922487 0.84 KDM1A (0.43) SIGMAR1KCNH2HDAC1PTGS2KDM1A
SCHEMBL28080410 0.75 SIGMAR1 (0.56) SIGMAR1KCNH2HDAC1PTGS2KDM1A
SCHEMBL755146 0.74 KDM5B (0.47)
SCHEMBL17961115 0.73 HDAC1 (0.51) SIGMAR1KCNH2HDAC1PTGS2KDM1A
SCHEMBL20644440 0.73 ESRRG (0.50) HDAC1NOTUMESRRG
SCHEMBL18460628 0.73 IDO1 (0.41) NOTUM
SCHEMBL20445146 0.73 IDO1 (0.41) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670247-B2 Contraceptive agents THE UNIVERSITY OF KANSAS (US) 2017-06-06 US disclosed