SCHEMBL28080410

SCHEMBL28080410

CNc1cn(Cc2ccc(F)cc2)nn1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.56
KCNH2 Q12809 1/20 0.55
HDAC1 Q13547 1/20 0.46
PTGS2 P35354 1/20 0.46
MAPT P10636 3/20 0.43
LMNA P02545 1/20 0.43
CDC7 O00311 1/20 0.42
ROCK2 O75116 1/20 0.42
GSK3B P49841 1/20 0.42
MAPK1 P28482 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM1A O60341 1/20 0.41
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27971447 0.83 SIGMAR1 (0.59) SIGMAR1LMNAGSK3BALDH1A1
SCHEMBL19611853 0.83 MEN1 (0.56) HDAC1PTGS2MAPTALDH1A1
SCHEMBL17961132 0.81 SIGMAR1 (0.51) SIGMAR1KCNH2HDAC1PTGS2MAPT
SCHEMBL28523893 0.79 SIGMAR1 (0.43) SIGMAR1KCNH2
SCHEMBL17961115 0.79 HDAC1 (0.51) SIGMAR1KCNH2HDAC1PTGS2MAPT
SCHEMBL9369847 0.76 CA5A (0.54) SIGMAR1KCNH2MAPTLMNAALDH1A1
SCHEMBL18925014 0.75 SIGMAR1 (0.45) SIGMAR1KCNH2HDAC1PTGS2MAPT
SCHEMBL28517969 0.75 SIGMAR1 (0.40) SIGMAR1KCNH2HDAC1
SCHEMBL17961139 0.75 MAPT (0.54) SIGMAR1KCNH2HDAC1PTGS2MAPT
SCHEMBL16401906 0.75 HDAC1 (0.49) SIGMAR1KCNH2HDAC1PTGS2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104059055-B 1,2, 3-triazole compound and preparation method and application thereof 常州大学 2016-08-31 CN disclosed
CN-105440020-A 1,2,3-triazole compounds with antitumor activity and preparation method for 1,2,3-triazole compounds UNIV CHANGZHOU 2016-03-30 CN disclosed
CN-104059055-A 1,2, 3-triazole compound and preparation method and application thereof UNIV CHANGZHOU 2014-09-24 CN disclosed