SCHEMBL1892896

SCHEMBL1892896

Cn1c(=O)[nH]c2c(ncn2-n2cnc3c(=O)[nH]c(=O)n(C)c32)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APAF1 O14727 1/20 0.39
CASP6 P55212 1/20 0.39
KDM4E B2RXH2 8/20 0.39
ALDH1A1 P00352 6/20 0.39
HPGD P15428 6/20 0.39
GAA P10253 2/20 0.39
GLA P06280 1/20 0.39
CYP3A4 P08684 2/20 0.38
PMP22 Q01453 2/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
BLM P54132 1/20 0.38
MAPK1 P28482 1/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
HSD17B10 Q99714 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7626818 0.88 CYP3A4 (0.46) APAF1CASP6KDM4EALDH1A1HPGD
SCHEMBL10947288 0.86 CYP3A4 (0.38) APAF1CASP6KDM4EALDH1A1HPGD
SCHEMBL4322373 0.75 CYP3A4 (0.54) APAF1CASP6KDM4EALDH1A1CYP3A4
SCHEMBL515776 0.75 ALDH1A1 (0.54) APAF1CASP6KDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL27932628 0.73 CYP3A4 (0.53) APAF1CASP6KDM4EALDH1A1HPGD
SCHEMBL27932684 0.72 CYP3A4 (0.44) APAF1CASP6KDM4EALDH1A1HPGD
SCHEMBL14879818 0.70 PMP22 (0.53) ALDH1A1GLACYP3A4PMP22MAPT
SCHEMBL17682322 0.69 CYP3A4 (0.41) APAF1CASP6KDM4EALDH1A1GAA
SCHEMBL28324506 0.69 LMNA (0.41) KDM4EALDH1A1CYP3A4PMP22LMNA
SCHEMBL7605281 0.69 CYP3A4 (0.41) APAF1CASP6KDM4EALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180251854-A1 Method For Predicting Therapy Responsiveness In Basal Like Tumors WIRTZ RALPH MARKUS (DE) 2018-09-06 US disclosed
US-9932639-B2 Method for predicting therapy responsiveness in basal like tumors WIRTZ RALPH MARKUS (DE) 2018-04-03 US disclosed
CN-102264235-A Food product fortified with methylxanthines 2011-11-30 CN disclosed
EP-2369939-A2 FOOD PRODUCTS ENRICHED WITH METHYLXANTHINES Unilever PLC (GB) 2011-10-05 EP disclosed
US-20110118129-A1 METHOD FOR PREDICTING THERAPY RESPONSIVENESS IN BASAL LIKE TUMORS Wirtz, Ralph Markus (DE) 2011-05-19 US disclosed
EP-2215251-A2 METHOD FOR PREDICTING THERAPY RESPONSIVENESS IN BASAL LIKE TUMORS Siemens Healthcare Diagnostics GmbH (DE) 2010-08-11 EP disclosed
WO-2010076112-A2 FOOD PRODUCTS ENRICHED WITH METHYLXANTHINES UNILEVER PLC (GB) 2010-07-08 WO disclosed
WO-2009068423-A2 METHOD FOR PREDICTING THERAPY RESPONSIVENESS IN BASAL LIKE TUMORS SIEMENS HEALTHCARE DIAGNOSTICS GMBH (DE) 2009-06-04 WO disclosed