SCHEMBL18937409

SCHEMBL18937409

CON(C)C(=O)c1cccc2cc[nH]c12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.57
PDPK1 O15530 1/20 0.55
BCHE P06276 3/20 0.51
MAPT P10636 3/20 0.45
KDM4E B2RXH2 2/20 0.45
RAB9A P51151 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GRM5 P41594 1/20 0.43
BACE1 P56817 1/20 0.42
KMT2A Q03164 2/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC2 Q92769 3/20 0.40
HDAC3 O15379 2/20 0.40
HDAC4 P56524 2/20 0.40
HDAC7 Q8WUI4 2/20 0.40
HDAC10 Q969S8 2/20 0.40
HDAC11 Q96DB2 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC9 Q9UKV0 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30088294 0.84 KEAP1 (0.64) KEAP1PDPK1BCHEMAPTKDM4E
SCHEMBL28600150 0.84 KEAP1 (0.64) KEAP1PDPK1BCHEMAPTKDM4E
SCHEMBL761721 0.78 KEAP1 (0.64) KEAP1PDPK1BCHEMAPTKDM4E
SCHEMBL30136593 0.78 KEAP1 (0.64) KEAP1PDPK1BCHEMAPTKDM4E
SCHEMBL5486616 0.77 KEAP1 (0.58) KEAP1PDPK1BCHEMAPTKDM4E
SCHEMBL8300350 0.77 KEAP1 (0.54) KEAP1PDPK1BCHEMAPTKDM4E
Hydrochloric Acid SCHEMBL28859534 0.76 KEAP1 (0.62) KEAP1PDPK1BCHEMAPTKDM4E
Hydrochloric Acid SCHEMBL7884796 0.75 PDPK1 (0.59) KEAP1PDPK1BCHEMAPTKDM4E
SCHEMBL3790885 0.75 KEAP1 (0.70) KEAP1PDPK1BCHEMAPTKDM4E
SCHEMBL30690400 0.75 KEAP1 (0.70) KEAP1PDPK1BCHEMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017093545-A1 ANTI-BACTERIAL COMPOUNDS BASED ON AMINO-GOLD PHOSPHINE COMPLEXES AUSPHERIX LIMITED (GB) 2017-06-08 WO disclosed