SCHEMBL18944162

SCHEMBL18944162

Cc1ccc(NCc2cnn(C)c2)c(C)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.44
MAPT P10636 1/20 0.44
GFER P55789 1/20 0.44
PDE10A Q9Y233 4/20 0.44
PDE1A P54750 7/20 0.43
PDE1B Q01064 7/20 0.43
PDE1C Q14123 7/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 1/20 0.43
BRD4 O60885 1/20 0.40
BRD9 Q9H8M2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31715868 0.74 PDE10A (0.45) PDE10APDE1APDE1BPDE1C
SCHEMBL18944430 0.73 MAPT (0.51) NPC1RAB9ASMN1; SMN2MAPTGFER
SCHEMBL29376709 0.73 PDE1A (0.43) SMN1; SMN2PDE10APDE1APDE1BPDE1C
SCHEMBL11175667 0.73 MAPT (0.61) NPC1RAB9ASMN1; SMN2MAPTGFER
SCHEMBL10557404 0.72 ALDH1A1 (0.74) RAB9ASMN1; SMN2MAPTKDM4EALDH1A1
SCHEMBL28736466 0.72 PDE1A (0.47) NPC1RAB9APDE10APDE1APDE1B
SCHEMBL31716208 0.71 HDAC8 (0.42) SMN1; SMN2GFERPDE10APDE1APDE1B
SCHEMBL28968809 0.70 KMT2A (0.58) SMN1; SMN2MAPTKDM4EALDH1A1GAA
SCHEMBL29120707 0.70 MCHR1 (0.62) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL31212184 0.70 LTA4H (0.49) NPC1RAB9ASMN1; SMN2PDE10APDE1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781661-B1 VASOPRESSIN V1A ANTAGONISTS VANTIA LTD (GB) 2017-06-07 EP disclosed