SCHEMBL18944310

SCHEMBL18944310

CCCCCCN1CCC(CC(=O)NCc2ccc(C(O)N3Cc4cnn(C)c4Nc4cc(C)ccc43)cc2F)CC1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 18/20 0.35
OXTR P30559 10/20 0.34
AVPR2 P30518 3/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM3 P20309 1/20 0.32
DRD3 P35462 1/20 0.32
OPRK1 P41145 1/20 0.32
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2129942 0.86 AVPR1A (0.48) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL18944344 0.78 P2RX7 (0.40) AVPR1AOXTRAVPR2
SCHEMBL18944343 0.77 AVPR1A (0.34) AVPR1AOXTRAVPR2
SCHEMBL2631700 0.75 AVPR1A (0.51) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL8266488 0.74 AVPR1A (0.52) AVPR1AOXTRAVPR2CHRM2CHRM4
Hydrochloric Acid SCHEMBL2129314 0.73 AVPR1A (0.51) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL18944341 0.72 AVPR1A (0.48) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2132179 0.70 AVPR1A (0.56) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2130284 0.70 AVPR1A (0.57) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2129541 0.69 AVPR1A (0.49) AVPR1AOXTRAVPR2CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781661-B1 VASOPRESSIN V1A ANTAGONISTS VANTIA LTD (GB) 2017-06-07 EP disclosed