SCHEMBL18944341

SCHEMBL18944341

Cc1cc(C(O)N2Cc3cnn(C)c3Nc3ccccc32)ccc1CNC(=O)CC1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 14/20 0.48
OXTR P30559 9/20 0.47
AVPR2 P30518 4/20 0.43
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRM3 P20309 1/20 0.43
DRD3 P35462 1/20 0.43
OPRK1 P41145 1/20 0.43
YAP1 P46937 3/20 0.36
TSPO P30536 1/20 0.36
GPR119 Q8TDV5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2130133 0.86 AVPR1A (0.67) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL18944306 0.84 AVPR1A (0.39) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL18944317 0.75 AVPR1A (0.47) AVPR1AOXTRAVPR2TSPO
SCHEMBL4832002 0.75 AVPR1A (0.81) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL18944305 0.75 AVPR1A (0.48) AVPR1AOXTRAVPR2TSPO
SCHEMBL2631711 0.74 AVPR1A (0.70) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL18944310 0.72 AVPR1A (0.35) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL2130151 0.72 AVPR1A (0.72) AVPR1AOXTRAVPR2CHRM2CHRM4
Hydrochloric Acid SCHEMBL2130197 0.72 AVPR1A (0.71) AVPR1AOXTRAVPR2CHRM2CHRM4
SCHEMBL1495942 0.71 TP53 (0.39) AVPR1AOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781661-B1 VASOPRESSIN V1A ANTAGONISTS VANTIA LTD (GB) 2017-06-07 EP disclosed