SCHEMBL18948426

SCHEMBL18948426

CCCCCCC(CCCCCC)c1nccnc1C

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.37
LMNA P02545 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
SLC2A1 P11166 1/20 0.32
DNM1 Q05193 1/20 0.31
GPR84 Q9NQS5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14155079 0.93 NR1I2 (0.42) NR1I2LMNAKDM4EHPGDSLC2A1
SCHEMBL19003645 0.84
SCHEMBL22770493 0.80 ADA (0.40) KDM4E
SCHEMBL21888617 0.77 FAAH (0.37) NR1I2LMNAKDM4E
SCHEMBL26041690 0.77 FAAH (0.37) NR1I2LMNAKDM4E
SCHEMBL22193276 0.76 HPGD (0.37) HPGD
SCHEMBL23491344 0.75 ADA (0.37) NR1I2GPR84
SCHEMBL26422953 0.75 SLC2A1 (0.31) NR1I2SLC2A1
SCHEMBL28377618 0.74 GPR84 (0.39) GPR84
SCHEMBL23870972 0.73 FAAH (0.36) NR1I2LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9676780-B2 Piperazine-substituted [1,2,4]triazolo[1,5-C]quinazolin-5-amine compounds with A2A antagonist properties MERCK SHARP & DOHME CORP. (US) 2017-06-13 US disclosed