SCHEMBL18975782

SCHEMBL18975782

CCC(CC)(CC#N)n1cc(-c2ccnc3[nH]ccc23)cn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 3/20 0.56
AURKA O14965 2/20 0.56
INCENP Q9NQS7 2/20 0.56
TPX2 Q9ULW0 2/20 0.56
JAK2 O60674 14/20 0.53
JAK1 P23458 9/20 0.53
JAK3 P52333 5/20 0.53
TYK2 P29597 2/20 0.53
GRM4 Q14833 1/20 0.49
CCNK O75909 2/20 0.44
CDK12 Q9NYV4 2/20 0.44
NUDT1 P36639 1/20 0.43
IKBKB O14920 1/20 0.42
CHUK O15111 1/20 0.42
DAPK3 O43293 1/20 0.42
PRKD3 O94806 1/20 0.42
MAP4K4 O95819 1/20 0.42
PAK4 O96013 1/20 0.42
CSF1R P07333 1/20 0.42
RET P07949 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL98899 0.83 JAK2 (0.56) AURKBAURKAJAK2JAK1JAK3
SCHEMBL99736 0.83 AURKB (0.56) AURKBAURKAINCENPTPX2JAK2
SCHEMBL21085376 0.82 AURKB (0.63) AURKBAURKAINCENPTPX2JAK2
SCHEMBL18602404 0.77 AURKB (0.57) AURKBAURKAINCENPTPX2JAK2
SCHEMBL99868 0.77 AURKB (0.59) AURKBAURKAINCENPTPX2JAK2
SCHEMBL19832104 0.77 AURKB (0.48) AURKBAURKAINCENPTPX2JAK2
SCHEMBL15389485 0.77 AURKB (0.56) AURKBAURKAINCENPTPX2JAK2
Trifluoroacetic Acid SCHEMBL99138 0.76 JAK2 (0.48) AURKBAURKAINCENPTPX2JAK2
Trifluoroacetic Acid SCHEMBL29541266 0.76 JAK2 (0.48) AURKBAURKAINCENPTPX2JAK2
SCHEMBL13541161 0.75 AURKB (0.63) AURKBAURKAINCENPTPX2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017097224-A1 AZETIDINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-15 WO disclosed