SCHEMBL19832104

SCHEMBL19832104

CCC(CCO)(CCNSC)n1cc(-c2ccnc3[nH]ccc23)cn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 2/20 0.48
AURKA O14965 1/20 0.48
INCENP Q9NQS7 1/20 0.48
TPX2 Q9ULW0 1/20 0.48
GRM4 Q14833 1/20 0.43
CCNK O75909 2/20 0.41
CDK12 Q9NYV4 2/20 0.41
NEK1 Q96PY6 5/20 0.40
JAK1 P23458 6/20 0.40
JAK2 O60674 5/20 0.40
JAK3 P52333 3/20 0.40
TYK2 P29597 1/20 0.40
NUDT1 P36639 1/20 0.39
IKBKB O14920 2/20 0.39
CHUK O15111 2/20 0.39
DAPK3 O43293 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
PAK4 O96013 1/20 0.39
CSF1R P07333 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99868 0.79 AURKB (0.59) AURKBAURKAINCENPTPX2GRM4
SCHEMBL18975782 0.77 AURKB (0.56) AURKBAURKAINCENPTPX2GRM4
SCHEMBL21085376 0.76 AURKB (0.63) AURKBAURKAINCENPTPX2GRM4
Trifluoroacetic Acid SCHEMBL99616 0.73 AURKB (0.51) AURKBAURKAINCENPTPX2GRM4
Trifluoroacetic Acid SCHEMBL29540674 0.73 AURKB (0.51) AURKBAURKAINCENPTPX2GRM4
SCHEMBL13774666 0.73 AURKB (0.62) AURKBAURKAINCENPTPX2GRM4
SCHEMBL15389485 0.73 AURKB (0.56) AURKBAURKAINCENPTPX2GRM4
SCHEMBL15389759 0.71 AURKB (0.54) AURKBAURKAINCENPTPX2GRM4
SCHEMBL100576 0.71 AURKB (0.62) AURKBAURKAINCENPTPX2GRM4
SCHEMBL98741 0.70 AURKA (0.55) AURKBAURKAINCENPTPX2GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018019222-A1 HETEROCYCLIC COMPOUND AS JAK INHIBITOR, AND SALTS AND THERAPEUTIC USE THEREOF 张文燕 2018-02-01 WO disclosed