SCHEMBL1897754

SCHEMBL1897754

O=C(CCc1ccc(F)cc1)Nc1scc(-c2ccc(Br)cc2)c1C(=O)OC(=O)c1c(-c2ccc(Br)cc2)csc1NC(=O)CCc1cccc(F)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
HTT P42858 4/20 0.49
MAPT P10636 4/20 0.49
LMNA P02545 3/20 0.49
NPSR1 Q6W5P4 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
TP53 P04637 3/20 0.47
KDM4E B2RXH2 3/20 0.46
RAB9A P51151 2/20 0.46
HPGD P15428 2/20 0.46
NPC1 O15118 1/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TDP1 Q9NUW8 2/20 0.42
POLB P06746 2/20 0.42
PTPN1 P18031 1/20 0.41
CASP3 P42574 2/20 0.40
SENP8 Q96LD8 2/20 0.40
SENP7 Q9BQF6 2/20 0.40
SENP6 Q9GZR1 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1897752 0.91 SMN1; SMN2 (0.52) ALDH1A1HTTMAPTLMNANPSR1
SCHEMBL1953935 0.87 CASP3 (0.53) ALDH1A1HTTMAPTLMNANPSR1
SCHEMBL1952338 0.83 SMN1; SMN2 (0.53) ALDH1A1HTTMAPTLMNANPSR1
SCHEMBL2776181 0.78 ANO1 (0.44) ALDH1A1HTTMAPTLMNANPSR1
SCHEMBL15241643 0.78 TP53 (0.46) ALDH1A1HTTSMN1; SMN2TP53RAB9A
SCHEMBL1953704 0.78 ANO1 (0.59) SMN1; SMN2TP53ANO1
SCHEMBL1954819 0.77 MEN1 (0.56) ALDH1A1HTTMAPTLMNANPSR1
SCHEMBL1952289 0.76 ANO1 (0.57) ALDH1A1HTTMAPTLMNANPSR1
SCHEMBL12271436 0.76 CASP3 (0.67) ALDH1A1HTTMAPTLMNANPSR1
SCHEMBL1951875 0.75 MEN1 (0.54) ALDH1A1HTTMAPTLMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321303-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2011-05-18 EP disclosed
WO-2010027875-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2010-03-11 WO disclosed