SCHEMBL1897771

SCHEMBL1897771

COc1ccc(OC)c(-c2ccc3c(c2)CC(=O)N3)c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 2/20 0.75
PDE3B Q13370 3/20 0.58
PDE3A Q14432 3/20 0.58
GRIA1 P42261 2/20 0.54
CACNG8 Q8WXS5 2/20 0.54
ABCB1 P08183 1/20 0.48
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
HDAC4 P56524 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
PGR P06401 1/20 0.46
BRD4 O60885 2/20 0.46
CREBBP Q92793 1/20 0.46
CYP1A2 P05177 2/20 0.45
CYP11B1 P15538 2/20 0.45
CYP11B2 P19099 2/20 0.45
SRC P12931 1/20 0.45
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10711490 0.90 TDP2 (0.75) TDP2PDE3BPDE3AMAOAMAOB
SCHEMBL18010814 0.86 TDP2 (1.00) TDP2PDE3BPDE3A
SCHEMBL155069 0.84 PDE3B (0.62) TDP2PDE3BPDE3AGRIA1CACNG8
SCHEMBL20214 0.83 PDE3B (0.66) TDP2PDE3BPDE3AGRIA1CACNG8
SCHEMBL31040124 0.83 PDE3B (0.66) TDP2PDE3BPDE3AGRIA1CACNG8
SCHEMBL4479338 0.79 TDP2 (0.64) TDP2PDE3BPDE3ABRD4CREBBP
SCHEMBL3285782 0.78 NPC1 (0.59) PDE3BPDE3AGRIA1CACNG8MAOA
SCHEMBL2170525 0.74 GRIA1 (0.49) TDP2PDE3BPDE3AGRIA1CACNG8
SCHEMBL10713385 0.74 PDE3B (0.55) TDP2PDE3BPDE3AMAOAMAOB
SCHEMBL1875842 0.74 CYP11B1 (0.79) PDE3BPDE3AGRIA1CACNG8PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed