SCHEMBL18979786

SCHEMBL18979786

Cc1c(NC(=O)c2ccncn2)cccc1-c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 9/20 0.55
ALDH1A1 P00352 2/20 0.54
TSHR P16473 2/20 0.54
ALOX15 P16050 1/20 0.54
PDCD1 Q15116 7/20 0.53
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
CHRNB2 P17787 1/20 0.51
CHRNB4 P30926 1/20 0.51
CHRNA3 P32297 1/20 0.51
CHRNA4 P43681 1/20 0.51
GSK3A P49840 3/20 0.47
GSK3B P49841 3/20 0.47
KDM4E B2RXH2 1/20 0.47
ATM Q13315 1/20 0.47
LMNA P02545 1/20 0.46
HSD17B10 Q99714 1/20 0.46
P2RX7 Q99572 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29516927 0.85 NPC1 (0.70) CD274ALDH1A1TSHRALOX15PDCD1
SCHEMBL18979807 0.84 ALDH1A1 (0.79) CD274ALDH1A1TSHRALOX15PDCD1
SCHEMBL18979851 0.81 PDCD1 (0.53) CD274ALDH1A1TSHRALOX15PDCD1
SCHEMBL22659481 0.80 NPC1 (0.51) CD274ALDH1A1NPC1RAB9AGSK3A
SCHEMBL18979779 0.80 NPC1 (0.51) CD274ALDH1A1TSHRALOX15PDCD1
SCHEMBL18979761 0.79 PDCD1 (0.59) CD274ALDH1A1TSHRALOX15PDCD1
SCHEMBL27965599 0.79 NPC1 (0.56) ALDH1A1NPC1RAB9AKDM4ELMNA
SCHEMBL18979774 0.79 CD274 (0.56) CD274ALDH1A1TSHRALOX15PDCD1
SCHEMBL18979867 0.78 PDCD1 (0.55) CD274ALDH1A1TSHRALOX15PDCD1
SCHEMBL13053955 0.78 NPC1 (0.62) CD274ALDH1A1PDCD1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260078113-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORP (US) 2026-03-19 US claimed
US-20180273519-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORPORATION 2018-09-27 US claimed
US-20170174671-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORPORATION 2017-06-22 US claimed
US-20260078113-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORP (US) 2026-03-19 US disclosed
US-12516044-B2 Heterocyclic compounds as immunomodulators INCYTE CORPORATION (US) 2026-01-06 US disclosed
EP-3390361-B1 N-PHENYL-PYRIDINE-2-CARBOXAMIDE DERIVATIVES AND THEIR USE AS PD-1/PD-L1 PROTEIN/PROTEIN INTERACTION MODULATORS INCYTE CORP (US) 2022-03-16 EP disclosed
EP-3390361-B1 N-PHENYL-PYRIDINE-2-CARBOXAMIDE DERIVATIVES AND THEIR USE AS PD-1/PD-L1 PROTEIN/PROTEIN INTERACTION MODULATORS INCYTE CORP (US) 2022-03-16 EP disclosed
US-20210363137-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORPORATION 2021-11-25 US disclosed
US-20210363137-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORPORATION 2021-11-25 US disclosed
US-20180273519-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORPORATION 2018-09-27 US disclosed
WO-2017106634-A1 N-PHENYL-PYRIDINE-2-CARBOXAMIDE DERIVATIVES AND THEIR USE AS PD-1/PD-L1 PROTEIN/PROTEIN INTERACTION MODULATORS INCYTE CORPORATION (US) 2017-06-22 WO disclosed
US-20170174671-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORPORATION 2017-06-22 US disclosed
US-20170174671-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS INCYTE CORPORATION 2017-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180273519-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS CD74, IL2, ICOS CD274 97/4885ALDH1A1 247/4885TSHR 2281/4885
US-20210363137-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS CD74, IL2, ICOS CD274 97/4885ALDH1A1 247/4885TSHR 2281/4885
US-20260078113-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS MSR1, NR3C1, CCR1 CD274 779/4885ALDH1A1 868/4885TSHR 113/4885
US-20170174671-A1 HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS CD74, IL2, ICOS CD274 97/4885ALDH1A1 247/4885TSHR 2281/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.