SCHEMBL1898425

SCHEMBL1898425

CC(C)n1cc(-c2ccccc2)[c]n1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.32
PTGS2 P35354 1/20 0.32
MAPT P10636 2/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 2/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
KMT2A Q03164 1/20 0.31
ATP1A1 P05023 4/20 0.30
ATP1B1 P05026 4/20 0.30
ATP1A3 P13637 4/20 0.30
ATP1B2 P14415 4/20 0.30
ATP1A2 P50993 4/20 0.30
ATP1B3 P54709 4/20 0.30
FXYD2 P54710 4/20 0.30
ATP1A4 Q13733 4/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL700238 0.75 PTGS2 (0.40) PTGS2MAPTLMNAHPGDMEN1
SCHEMBL1851644 0.75 KMT2A (0.41) MAPTHPGDMEN1ALDH1A1KMT2A
SCHEMBL1902680 0.70 KMT2A (0.34) MAPTHPGDMEN1ALDH1A1GLA
SCHEMBL1900677 0.70 L3MBTL1 (0.36) CYP19A1MAPTLMNAHPGDALDH1A1
SCHEMBL16911497 0.66
SCHEMBL16912032 0.66
SCHEMBL13322631 0.65 CREBBP (0.48) MAPTLMNA
SCHEMBL9963176 0.64 CYP19A1 (0.66) CYP19A1PTGS2LMNAMEN1GAA
SCHEMBL19088674 0.64 PDE1A (0.45) PTGS2MAPTHPGDMEN1ALDH1A1
SCHEMBL23399527 0.63 KMT2A (0.43) PTGS2MAPTLMNAHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8455477-B2 Therapeutic compounds MERCK SHARP & DOHME CORP. (US) 2013-06-04 US disclosed
US-20110207711-A1 Therapeutic Compounds MSD K.K. (JP) 2011-08-25 US disclosed
EP-2320907-A1 THERAPEUTIC COMPOUNDS Merck & Co., Inc. (US) 2011-05-18 EP disclosed
WO-2010017047-A1 THERAPEUTIC COMPOUNDS MERCK & CO., INC. (US) 2010-02-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110207711-A1 Therapeutic Compounds WEE2, MARK3, WEE1 CYP19A1 3806/4885PTGS2 4337/4885MAPT 90/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.