SCHEMBL1898665

SCHEMBL1898665

NC(=O)c1ccccc1-c1ccccc1Br

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.59
METAP2 P50579 1/20 0.50
GRM2 Q14416 1/20 0.49
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 2/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
CSNK1A1 P48729 1/20 0.46
TYRO3 Q06418 1/20 0.46
DYRK1B Q9Y463 1/20 0.46
RAB9A P51151 3/20 0.46
POLB P06746 2/20 0.46
KMT2A Q03164 2/20 0.45
NUDT1 P36639 1/20 0.44
CHEK1 O14757 1/20 0.43
NPC1 O15118 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29941064 1.00 BCAT2 (0.59) BCAT2METAP2GRM2KDM4EALDH1A1
SCHEMBL30514077 0.87 BCAT2 (0.74) BCAT2METAP2KDM4EALDH1A1MAPT
SCHEMBL210767 0.87 BCAT2 (0.74) BCAT2METAP2KDM4EALDH1A1MAPT
SCHEMBL15952999 0.86 BCAT2 (0.53) BCAT2METAP2GRM2KDM4EALDH1A1
Hydrochloric Acid SCHEMBL16463881 0.84 BCAT2 (0.71) BCAT2METAP2KDM4EALDH1A1MAPT
SCHEMBL1110181 0.84 BCAT2 (0.71) BCAT2METAP2KDM4EALDH1A1MAPT
SCHEMBL31012518 0.84 BCAT2 (0.71) BCAT2METAP2KDM4EALDH1A1MAPT
SCHEMBL27704996 0.84 KEAP1 (0.58) BCAT2METAP2GRM2KDM4EALDH1A1
SCHEMBL28368379 0.83 KMT2A (0.47) GRM2ALDH1A1MAPTTSHRRAB9A
SCHEMBL1898663 0.82 KEAP1 (0.56) BCAT2METAP2KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103553859-B A kind of method being prepared aminated compounds intermediate by acid amides DU YEHONG (CN) 2015-09-16 CN disclosed
CN-103553859-A Method for preparing amine compound midbody by utilizing amide ZHU YEHONG 2014-02-05 CN disclosed
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed
WO-2003076930-A1 METHOD FOR CHARACTERIZING METABOLITES USING HYDROGEN/DEUTERIUM EXCHANGE WARNER-LAMBERT COMPANY LLC (US) 2003-09-18 WO disclosed
US-20030175979-A1 System and method for characterizing metabolites using hydrogen/deuterium exchange LAM WING WAH (US) 2003-09-18 US disclosed
EP-1345028-A1 Method for charcterizing metabolites using hydrogen/deuterium exchange Warner-Lambert Company LLC (US) 2003-09-17 EP disclosed