SCHEMBL18995019

SCHEMBL18995019

CCc1ccc(OC)c(-n2nnnc2C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 3/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 9/20 0.41
TSHR P16473 5/20 0.41
LMNA P02545 4/20 0.41
HTT P42858 4/20 0.41
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KCNN4 O15554 2/20 0.41
RAB9A P51151 3/20 0.41
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
NPC1 O15118 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
PKM P14618 1/20 0.38
STAT3 P40763 1/20 0.38
KMT2A Q03164 1/20 0.38
GALR3 O60755 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15786417 0.82 KMT2A (0.55) NR1I2USP2ALDH1A1TSHRLMNA
SCHEMBL18994950 0.79 LMNA (0.44) LMNAKCNN4NPC1
SCHEMBL15783484 0.77 NR1I2 (0.55) NR1I2
SCHEMBL19836576 0.77 NR1I2 (0.42) NR1I2USP2ALDH1A1TSHRLMNA
SCHEMBL4203800 0.77 ATM (0.55) USP2ALDH1A1TSHRMAPTTP53
SCHEMBL4211677 0.75 KCNN4 (0.66) NR1I2ALDH1A1TSHRLMNAHTT
SCHEMBL17550642 0.72 LMNA (0.43) ALDH1A1TSHRLMNAHTTMAPT
SCHEMBL18066884 0.72 LRRK2 (0.39) USP2ALDH1A1TSHRLMNAHTT
SCHEMBL10066944 0.72 LMNA (0.64) ALDH1A1LMNAHTTMAPTTP53
SCHEMBL17708385 0.69 LRRK2 (0.43) USP2ALDH1A1TSHRLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9682976-B2 Protein kinase C inhibitors and uses thereof RIGEL PHARMACEUTICALS, INC. (US) 2017-06-20 US disclosed