SCHEMBL189981

SCHEMBL189981

COC(=O)C1CSCC1=O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
BRD4 O60885 1/20 0.34
CYP1A2 P05177 2/20 0.33
HIF1A Q16665 1/20 0.33
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 2/20 0.31
HSD17B10 Q99714 1/20 0.31
MMP2 P08253 1/20 0.31
ANPEP P15144 1/20 0.31
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10267038 0.81 CYP1A2 (0.34) KMT2ABRD4CYP1A2HIF1AALDH1A1
SCHEMBL2904103 0.81 KMT2A (0.36) KMT2ABRD4CYP1A2HIF1AALDH1A1
SCHEMBL172419 0.79 ALDH1A1 (0.45) KMT2AALDH1A1KDM4EHSD17B10HPGD
SCHEMBL7783338 0.78 KMT2A (0.34) KMT2ABRD4
SCHEMBL4703163 0.77 ALDH1A1 (0.43) KMT2AALDH1A1HSD17B10
SCHEMBL10362738 0.77 ALDH1A1 (0.43) KMT2AALDH1A1HSD17B10
SCHEMBL4703164 0.77 ALDH1A1 (0.43) KMT2AALDH1A1HSD17B10
SCHEMBL28798717 0.76 KMT2A (0.32) KMT2A
SCHEMBL9511588 0.74 L3MBTL1 (0.39) CYP1A2ALDH1A1KDM4EHPGDCYP2C19
SCHEMBL10423608 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 325 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0344983-B1 PROCESS FOR PREPARING 2- AND 4-ALKOXYCARBONYL THIOLAN-3-ONES JOHN WYETH & BROTHER LIMITED (GB) 1993-09-15 EP claimed
EP-0344983-A1 Process for preparing 2- and 4-alkoxycarbonyl thiolan-3-ones JOHN WYETH & BROTHER LIMITED (GB) 1989-12-06 EP claimed
EP-4339199-B1 SYNTHESIS OF CANTHARIDIN VERRICA PHARMACEUTICALS INC (US) 2026-05-20 EP disclosed
EP-3901151-B1 HALOGENATED-HETEROARYL AND OTHER HETEROCYCLIC KINASE INHIBITORS, AND USES THEREOF IOMX THERAPEUTICS AG (DE) 2026-04-01 EP disclosed
US-20250296928-A1 A SYNTHESIS SCHEME AND PROCEDURES FOR PREPARING A SIK3 INHIBITOR AND INTERMEDIATES THEREOF IOMX THERAPEUTICS AG (DE) 2025-09-25 US disclosed
WO-2025119351-A1 GPR139 AGONIST 深圳湾实验室 2025-06-12 WO disclosed
CN-120035585-A Process for the preparation of substituted aminothiophenes 安道麦阿甘有限公司 2025-05-23 CN disclosed
US-20250115604-A1 SULFOXIMINE GLYCOSIDASE INHIBITORS ASCENEURON SA (CH) 2025-04-10 US disclosed
US-20250100966-A1 MEK INHIBITORS AND METHODS OF THEIR USE EXELIXIS INC (US) 2025-03-27 US disclosed
CN-116265451-B Preparation method of 4-methoxycarbonyl-2-methylthiophene-3-sulfonamide 江苏瑞邦农化股份有限公司 2025-02-14 CN disclosed
US-12221452-B2 Synthesis of cantharidin VERRICA PHARMACEUTICALS INC. (US) 2025-02-11 US disclosed
US-4144235-A ANTIPSYCHOTIC, NEUROLEPTIC AMERICAN CYANAMID COMPANY (US) 1979-03-13 US disclosed
US-4087421-A NEUROLEPTIC, ANTI-DEPRESSANT AND ANALGESTIC ACTIVITY AMERICAN CYANAMID COMPANY (US) 1978-05-02 US disclosed
US-4025630-A Anesthesia methods using benzopyrans and esters thereof as pre-anesthesia medication ABBOTT LABORATORIES (US) 1977-05-24 US disclosed
US-4007272-A Substituted benzodiazepin-10-ones in treating pain and depression AMERICAN CYANAMID COMPANY (US) 1977-02-08 US disclosed
US-3972880-A TRANQUILIZER SHARPS ASSOCIATES (US) 1976-08-03 US disclosed
US-3960871-A ANTIDEPRESSANT, ANALGESICS, ANTICONVULSANT ANTI-ANXIETY ACTIVITY SHARPS ASSOCIATES (US) 1976-06-01 US disclosed
US-3953430-A ANTIDEPRESSANTS, ANALGESICS AMERICAN CYANAMID COMPANY (US) 1976-04-27 US disclosed
US-3951981-A NEUROLEPTIC, ANALGESIC AMERICAN CYANAMID COMPANY (US) 1976-04-20 US disclosed
US-3940421-A Intermediates for the preparation of thienobenzopyrans and thiopyranobenzopyrans ARTHUR D. LITTLE, INC. (US) 1976-02-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250115604-A1 SULFOXIMINE GLYCOSIDASE INHIBITORS ENGASE, BACE1, GAA KMT2A 973/4885BRD4 4319/4885CYP1A2 1194/4885
US-20250100966-A1 MEK INHIBITORS AND METHODS OF THEIR USE BRAF, NRAS, KRAS KMT2A 1630/4885BRD4 1308/4885CYP1A2 1217/4885
US-12221452-B2 Synthesis of cantharidin TYR, CMA1, DPM1 KMT2A 4610/4885BRD4 449/4885CYP1A2 239/4885
US-20250296928-A1 A SYNTHESIS SCHEME AND PROCEDURES FOR PREPARING A SIK3 INHIBITOR AND INTERMEDIATES THEREOF SIK3, SIK1, SIK2 KMT2A 2822/4885BRD4 1284/4885CYP1A2 2310/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.