SCHEMBL1900222

SCHEMBL1900222

Cc1ccc(-c2nc(N)c3cc[nH]c3n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 3/20 0.53
CYP1A2 P05177 3/20 0.53
CYP1B1 Q16678 3/20 0.53
DPP4 P27487 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ADORA1 P30542 3/20 0.39
RAB9A P51151 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 1/20 0.39
GLA P06280 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
DYRK1A Q13627 1/20 0.39
HPGD P15428 1/20 0.39
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
ADORA3 P0DMS8 2/20 0.38
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14274543 0.83 ADORA1 (0.51) CYP1A1CYP1A2CYP1B1DPP4ADORA1
SCHEMBL7661563 0.81 ADORA1 (0.39) CYP1A1CYP1A2CYP1B1NPSR1ADORA1
SCHEMBL30165634 0.77 ADORA2A (0.47) ADORA1NPC1ADORA2A
SCHEMBL29981526 0.75 DYRK1A (0.46) ADORA1DYRK1AIKBKBCHUKHRH4
SCHEMBL18055932 0.75 DYRK1A (0.46) ADORA1DYRK1AIKBKBCHUKHRH4
SCHEMBL16826600 0.75 AURKA (0.52) ADORA1HRH4ADORA3
Hydrochloric Acid SCHEMBL29616498 0.74 DYRK1A (0.44) ADORA1DYRK1AIKBKBCHUKHRH4
Hydrochloric Acid SCHEMBL29616579 0.74 DYRK1A (0.44) ADORA1DYRK1AIKBKBCHUKHRH4
SCHEMBL16497095 0.73 NUDT1 (0.43) ADORA1DYRK1AIKBKBCHUKHRH4
SCHEMBL30110740 0.73 EGFR (0.53) CYP1A1CYP1A2CYP1B1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011060440-A2 KINASE INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-05-19 WO disclosed