SCHEMBL1900349

SCHEMBL1900349

CCC(c1ccc(N=C=O)cc1)c1ccc(N=C=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.50
TSHR P16473 1/20 0.50
TRPA1 O75762 1/20 0.40
GABRA1 P14867 1/20 0.38
GABRB2 P47870 1/20 0.38
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP1A2 P05177 1/20 0.38
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
CYP17A1 P05093 3/20 0.34
CYP2C9 P11712 2/20 0.32
MIF P14174 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10441237 0.90 CYP3A4 (0.42) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL3842072 0.82 CYP2C9 (0.49) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL9185663 0.79 CYP3A4 (0.46) CYP3A4TSHRTRPA1GABRA1GABRB2
Butane SCHEMBL16872374 0.78 CYP3A4 (0.62) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL30295346 0.77 CYP3A4 (0.50) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL14289853 0.77 ALDH1A1 (0.41) CYP3A4TSHRMAPK1TDP1CYP1A2
SCHEMBL131853 0.77 CYP3A4 (0.50) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL141743 0.77 CYP3A4 (0.50) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL9178584 0.77 CYP3A4 (0.43) CYP3A4TSHRTRPA1GABRA1GABRB2
SCHEMBL93536 0.76 CYP3A4 (0.54) CYP3A4TSHRTRPA1GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 132 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6593444-B2 Based on poly(1,3-propanediol carbonate) diol; hardness, higher elasticity modulus, and improved softening temperature and coefficient of thermal expansion; clarity; mechanical properties; extrusion SHELL OIL COMPANY 2003-07-15 US claimed
US-20020052461-A1 Thermoplastic polyurethane elastomers (TPUs) prepared with polytrimethylene carbonate soft segment SHELL OIL COMPANY 2002-05-02 US claimed
EP-0361122-A2 Rounding of hard cover books National Starch and Chemical Investment Holding Corporation (US) 1990-04-04 EP claimed
US-4342860-A AN UNSATUREATED IMIDE IS USED WITH A DI OR POLYISOCYANATE TO FORM A POLYIMIDE POLYMER RHONE-POULENC INDUSTRIES (FR) 1982-08-03 US claimed
US-4342861-A AN UNSATURATGED IMIDE AND A DI OR POLYISOCYANATE GO TO MAKE UP A POLYIMIDE POLYMER WHICH ALSO CONTAINS REPEATING AMIDE GROUPS RHONE-POULENC INDUSTRIES (FR) 1982-08-03 US claimed
US-4302572-A MOLDING MATERIALS; COATINGS; HEAT RESISTANCE; THIN FILMS RHONE-POULENC INDUSTRIES (FR) 1981-11-24 US claimed
US-20240157505-A1 POLISHING PAD UNIVERSAL PHOTONICS FAR EAST INC. (JP) 2024-05-16 US disclosed
WO-2024074778-A1 TWO-COMPONENT COMPOSITION COMPRISING AN ORGANOBORANE AMINE COMPLEX BOSTIK SA (FR) 2024-04-11 WO disclosed
EP-2912105-B1 DEFORMABLE FILM BENECKE KALIKO AG (DE) 2024-03-20 EP disclosed
EP-3999558-B1 TWO-COMPONENT ADHESIVE COMPOSITION COMPRISING A BORANE-AMINE COMPLEX BOSTIK SA (FR) 2023-11-22 EP disclosed
CN-116669903-A Polishing pad 美国环球光学有限公司 2023-08-29 CN disclosed
EP-3999579-B1 TWO-COMPONENT ADHESIVE COMPOSITION COMPRISING AN ORGANOBORANE AMINE COMPLEX BOSTIK SA (FR) 2023-06-28 EP disclosed
CN-115233331-A Bio-based spandex fiber and preparation method thereof 连云港杜钟新奥神氨纶有限公司 2022-10-25 CN disclosed
US-4187365-A FROM POLYISOCYANATE, FORMIC ACID, AND DICARBOXYLIC ANHYDRIDE CONTAINING ANOTHER ACID GROUP BAYER AKTIENGESELLSCHAFT (DE) 1980-02-05 US disclosed
US-4143060-A REACTING AN ISOCYANATO- SUBSTITUTED SILAIMIDAZOLIDONE DERIVATIVE WITH A URETHANE CONTAINING POLYMER BAYER AKTIENGESELLSCHAFT (DE) 1979-03-06 US disclosed
US-4088637-A Process for the production of polycondensates containing imide groups BAYER AKTIENGESELLSCHAFT (DT) 1978-05-09 US disclosed
US-4085165-A ISOCYANATE PREPOLYMER, VINYL COMPOUND, POLYAMINE OR POLYETHER CURING AGENT BRIDGESTONE TIRE CO., LTD. (JA) 1978-04-18 US disclosed
US-4062825-A SILICA BRIDGESTONE TIRE COMPANY, LTD. (JA) 1977-12-13 US disclosed
US-4018967-A POLYPHOSPHONITRILES AS LUBRICANTS BASF AKTIENGESELLSCHAFT (DT) 1977-04-19 US disclosed
US-3993641-A Process for the production of polyisocyanates containing uretdione groups BAYER AKTIENGESELLSCHAFT (DT) 1976-11-23 US disclosed