SCHEMBL19004850

SCHEMBL19004850

Nc1cc(N2CC(C(F)(F)F)C2)ncn1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.42
CA2 P00918 1/20 0.42
CHKA P35790 1/20 0.42
RPS6KB1 P23443 6/20 0.37
AKT1 P31749 5/20 0.36
RIPK1 Q13546 1/20 0.36
BTK Q06187 2/20 0.34
DPP4 P27487 5/20 0.33
MBOAT4 Q96T53 1/20 0.33
ACACB O00763 1/20 0.32
DPP8 Q6V1X1 1/20 0.32
DPP7 Q9UHL4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6119348 0.84 AKT1 (0.38) CA2CHKARPS6KB1AKT1RIPK1
SCHEMBL24027079 0.80 PSEN1 (0.39) MAP4K4ACACB
SCHEMBL26975070 0.77 AKT1 (0.38) MAP4K4CA2CHKARPS6KB1AKT1
SCHEMBL792633 0.77 EGLN2 (0.40) CA2CHKARPS6KB1AKT1RIPK1
SCHEMBL10187294 0.75 SMPD3 (0.41) RPS6KB1AKT1RIPK1BTKDPP4
SCHEMBL10187281 0.73 LRRK2 (0.42) MAP4K4AKT1DPP4
SCHEMBL23294851 0.73 LRRK2 (0.41) RPS6KB1AKT1RIPK1BTKDPP4
SCHEMBL12650637 0.73 HRH3 (0.51) BTK
SCHEMBL23024963 0.72 BTK (0.36) RPS6KB1AKT1RIPK1BTKDPP4
SCHEMBL20732640 0.71 SORD (0.41) MAP4K4RIPK1DPP4DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102091-A1 HETEROARYLBENZIMIDAZOLE COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-22 WO disclosed