SCHEMBL19005013

SCHEMBL19005013

Cc1ccnc(OC(C)C)c1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.49
NOS3 P29474 3/20 0.43
NOS2 P35228 3/20 0.43
HTR6 P50406 3/20 0.36
CCR1 P32246 1/20 0.35
CCR5 P51681 1/20 0.35
CCR8 P51685 1/20 0.35
ALOX5AP P20292 2/20 0.33
FEN1 P39748 2/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
PSMD14 O00487 1/20 0.32
COPS5 Q92905 1/20 0.32
SSTR4 P31391 1/20 0.32
SLC13A5 Q86YT5 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MKNK2 Q9HBH9 2/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
CDK1 P06493 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18985784 0.80 LRRK2 (0.46) LRRK2HTR6ALOX5APFEN1TRPM8
SCHEMBL27727585 0.80 NOS2 (0.50) LRRK2NOS3NOS2CCR1CCR5
SCHEMBL25411688 0.80 LRRK2 (0.46) LRRK2HTR6ALOX5APFEN1TRPM8
SCHEMBL3562229 0.80 LRRK2 (0.46) LRRK2NOS3NOS2CCR1CCR5
SCHEMBL6792963 0.76 NOS3 (0.48) LRRK2NOS3NOS2CCR1CCR5
SCHEMBL2614923 0.75 LRRK2 (0.45) LRRK2NOS3NOS2ALOX5APFEN1
SCHEMBL29497424 0.75 LRRK2 (0.45) LRRK2NOS3NOS2ALOX5APFEN1
SCHEMBL16231386 0.72 HPGD (0.50) LRRK2NOS3NOS2CCR1CCR5
SCHEMBL13409373 0.72 CYP1A2 (0.45) LRRK2CCR1CCR5CCR8ALOX5AP
SCHEMBL8382615 0.71 LRRK2 (0.44) LRRK2ALOX5APFEN1TRPM8SLC13A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102091-A1 HETEROARYLBENZIMIDAZOLE COMPOUNDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-06-22 WO disclosed