SCHEMBL19006668

SCHEMBL19006668

C=C(C)CC(C)[C@@H]1N=C(c2ccccn2)c2cc(Br)ccc2-n2c(C)cnc21

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.43
GABRA5 P31644 3/20 0.43
GABRA2 P47869 3/20 0.43
GABRB2 P47870 3/20 0.43
GABRA3 P34903 2/20 0.43
CHRM1 P11229 1/20 0.32
ADRA1A P35348 1/20 0.31
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5772396 0.90 GABRA1 (0.43) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL19006662 0.88 GABRA1 (0.42) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL19006536 0.88 GABRA1 (0.42) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL11824906 0.80 GABRA5 (0.51) GABRA1GABRA5GABRA2GABRB2GABRA3
Acetic Acid SCHEMBL11828455 0.78 GABRA1 (0.47) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL20545137 0.78 CHRM1 (0.42) CHRM1
SCHEMBL20473291 0.78 CHRM1 (0.42) CHRM1
SCHEMBL19006552 0.78 CHRM1 (0.42) CHRM1
SCHEMBL5769443 0.78 GABRA1 (0.43) GABRA1GABRA5GABRA2GABRB2GABRA3
SCHEMBL14328999 0.77 GABRA5 (0.48) GABRA1GABRA5GABRA2GABRB2GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017101808-A1 SHORT-ACTING BENZODIAZEPINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed