SCHEMBL19006935

SCHEMBL19006935

Cc1cc(C)cc(N(C)CCN(C)C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 8/20 0.41
NOS3 P29474 7/20 0.39
NOS2 P35228 5/20 0.39
HRH3 Q9Y5N1 1/20 0.33
CA12 O43570 1/20 0.33
CA2 P00918 1/20 0.33
CA3 P07451 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
ALDH1A1 P00352 4/20 0.32
TSHR P16473 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
TSPO P30536 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22607273 0.82 NOS1 (0.35) NOS1NOS3NOS2ALDH1A1CYP1A2
SCHEMBL10104262 0.81 NOS1 (0.45) NOS1NOS3NOS2TSHRCYP1A2
SCHEMBL10712858 0.79 ALDH1A1 (0.39) ALDH1A1TSPOKDM4E
SCHEMBL11056074 0.79 MAPT (0.36) NOS1NOS3NOS2ALDH1A1TSHR
SCHEMBL13959882 0.78 NOS1 (0.33) NOS1NOS3NOS2
SCHEMBL10104346 0.77 MCHR1 (0.36) NOS1NOS3NOS2
SCHEMBL17345678 0.77 NOS1 (0.37) NOS1NOS3NOS2HRH3ALDH1A1
SCHEMBL14174805 0.76 ALDH1A1 (0.50) NOS1HRH3CA12CA2CA9
SCHEMBL10104385 0.76 CYP2D6 (0.33) NOS1NOS2CYP2D6
SCHEMBL11121102 0.76 HPGD (0.36) NOS1NOS3NOS2ALDH1A1TSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170174689-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS VANDERBILT UNIVERSITY 2017-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170174689-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS MCL1, BCL2L1, BCL3 NOS1 1520/4885NOS3 2136/4885NOS2 1536/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.