SCHEMBL19013262

SCHEMBL19013262

CC(C)(C)OC(=O)n1c(C(=O)O)cc2ccc(Cl)cc21

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR9 P51686 7/20 0.51
CCR2 P41597 6/20 0.44
AURKA O14965 1/20 0.41
CDK2 P24941 1/20 0.41
NR1H2 P55055 5/20 0.39
NR1H3 Q13133 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18989603 0.87 PTGS2 (0.43) CCR9AURKACDK2NR1H2
SCHEMBL29632037 0.87 PTGS2 (0.43) CCR9AURKACDK2NR1H2
SCHEMBL17022491 0.83 NR1H2 (0.40) CCR9NR1H2NR1H3MEN1KMT2A
SCHEMBL13515283 0.83 AKR1C3 (0.40) CCR9NR1H2NR1H3MEN1KMT2A
SCHEMBL19013264 0.83 CCR9 (0.39) CCR9NR1H2NR1H3MEN1KMT2A
SCHEMBL28106960 0.82 NR1H2 (0.39) CCR9NR1H2NR1H3MEN1KMT2A
SCHEMBL29781083 0.82 NR1H2 (0.55) NR1H2NR1H3
SCHEMBL7902953 0.82 NR1H2 (0.55) NR1H2NR1H3
SCHEMBL17220641 0.81 NR1H2 (0.58) NR1H2NR1H3
SCHEMBL18989952 0.80 NR1H2 (0.41) CCR9NR1H2NR1H3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017106352-A1 CAFFEINE INHIBITORS OF MTHFD2 AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2017-06-22 WO disclosed