SCHEMBL1901384

SCHEMBL1901384

Nc1ccc(CNC(=O)[C@H](Cc2cccc3ccccc23)NC(=O)Cc2ccccc2F)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.46
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 1/20 0.44
OPRD1 P41143 1/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 1/20 0.43
PIN1 Q13526 1/20 0.42
LCK P06239 2/20 0.42
PSMB8 P28062 1/20 0.42
PSMB5 P28074 1/20 0.42
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA4 P43681 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRM1 Q13255 1/20 0.41
FURIN P09958 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1901386 1.00 MCHR1 (0.46) MCHR1KDM4EALDH1A1OPRD1KMT2A
SCHEMBL1905796 0.91 HTT (0.43) MCHR1KDM4EALDH1A1OPRD1KMT2A
SCHEMBL1905797 0.91 HTT (0.43) MCHR1KDM4EALDH1A1OPRD1KMT2A
SCHEMBL1902805 0.90 OPRD1 (0.46) MCHR1OPRD1PIN1LCKPSMB8
SCHEMBL1902802 0.90 OPRD1 (0.46) MCHR1OPRD1PIN1LCKPSMB8
SCHEMBL1906667 0.89 MCHR1 (0.44) MCHR1ALDH1A1OPRD1KMT2AMEN1
SCHEMBL1901459 0.89 OPRD1 (0.45) MCHR1OPRD1LCKPSMB8PSMB5
SCHEMBL1906669 0.89 MCHR1 (0.44) MCHR1ALDH1A1OPRD1KMT2AMEN1
SCHEMBL1904628 0.88 MCHR1 (0.50) MCHR1OPRD1LCKPSMB5FURIN
SCHEMBL1906797 0.88 OPRD1 (0.47) MCHR1OPRD1LCKPSMB8PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011051671-A1 AMINOPYRIDINE DERIVATIVES AS KALLIKREIN INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO claimed
WO-2011051671-A1 AMINOPYRIDINE DERIVATIVES AS KALLIKREIN INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO disclosed