SCHEMBL1902805

SCHEMBL1902805

Nc1ccc(CNC(=O)C(Cc2cccc3ccccc23)NC(=O)Cc2ccccc2O)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.46
MCHR1 Q99705 1/20 0.45
LCK P06239 3/20 0.44
FURIN P09958 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
MASP2 O00187 1/20 0.41
HRH4 Q9H3N8 1/20 0.40
MME P08473 1/20 0.40
ACE P12821 1/20 0.40
CPA1 P15085 1/20 0.40
ACE2 Q9BYF1 1/20 0.40
PSMB8 P28062 1/20 0.39
PSMB5 P28074 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1902802 1.00 OPRD1 (0.46) OPRD1MCHR1LCKFURINCTSS
SCHEMBL1901386 0.90 MCHR1 (0.46) OPRD1MCHR1LCKFURINCTSS
SCHEMBL1906667 0.90 MCHR1 (0.44) OPRD1MCHR1LCKFURINCTSS
SCHEMBL1906669 0.90 MCHR1 (0.44) OPRD1MCHR1LCKFURINCTSS
SCHEMBL1901384 0.90 MCHR1 (0.46) OPRD1MCHR1LCKFURINCTSS
SCHEMBL1901459 0.90 OPRD1 (0.45) OPRD1MCHR1LCKFURINCTSS
SCHEMBL1906797 0.89 OPRD1 (0.47) OPRD1MCHR1LCKCTSSCTSK
SCHEMBL1906792 0.89 OPRD1 (0.47) OPRD1MCHR1LCKCTSSCTSK
SCHEMBL1904628 0.87 MCHR1 (0.50) OPRD1MCHR1LCKFURINCTSS
SCHEMBL1904838 0.87 TACR1 (0.44) OPRD1MCHR1LCKFURINCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011051671-A1 AMINOPYRIDINE DERIVATIVES AS KALLIKREIN INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO claimed
WO-2011051671-A1 AMINOPYRIDINE DERIVATIVES AS KALLIKREIN INHIBITORS VANTIA LIMITED (GB) 2011-05-05 WO disclosed