SCHEMBL19014091

SCHEMBL19014091

O=C(CCC(F)(F)F)N1CC2CCC(C1)N2I

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.37
NPC1 O15118 1/20 0.36
NAMPT P43490 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19013670 0.90 EPHX2 (0.34) EPHX2NPC1NAMPT
SCHEMBL19013719 0.83 NPC1 (0.39) EPHX2NPC1
SCHEMBL20682211 0.81 NPC1 (0.40) EPHX2NPC1
SCHEMBL19013649 0.81 NPC1 (0.38) EPHX2NPC1
SCHEMBL19013705 0.80 NPC1 (0.37) EPHX2NPC1
SCHEMBL20743075 0.77 EPHX2 (0.39) EPHX2NPC1
SCHEMBL19014058 0.77 EPHX2 (0.32) EPHX2NPC1
SCHEMBL20743113 0.75 MEN1 (0.48) EPHX2
SCHEMBL31655313 0.75 EPHX2 (0.37) EPHX2NPC1
SCHEMBL20743046 0.75 ALDH1A1 (0.39) EPHX2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017103188-A1 THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-06-22 WO disclosed