SCHEMBL19013670

SCHEMBL19013670

O=C(CCC(F)(F)F)N1CC2CC(C1)N2I

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
CHRNB3 Q05901 1/20 0.34
CHRNA6 Q15825 1/20 0.34
NPC1 O15118 2/20 0.34
NAMPT P43490 1/20 0.34
CCR2 P41597 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19014091 0.90 EPHX2 (0.37) EPHX2NPC1NAMPT
SCHEMBL20682275 0.81 CHRNB2 (0.36) EPHX2CHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL19014100 0.77 CCR2 (0.33) CCR2
SCHEMBL19013719 0.77 NPC1 (0.39) EPHX2NPC1
SCHEMBL14211346 0.76 CHRNB2 (0.61) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL20743113 0.75 MEN1 (0.48) EPHX2
SCHEMBL31655313 0.75 EPHX2 (0.37) EPHX2CHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL20682211 0.74 NPC1 (0.40) EPHX2NPC1
SCHEMBL19013649 0.74 NPC1 (0.38) EPHX2CHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL19014535 0.74 CCR2 (0.43) CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017103188-A1 THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-06-22 WO disclosed