SCHEMBL19014100

SCHEMBL19014100

O=C(CCC(F)(F)F)N1C2CC1CN(I)C2

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 2/20 0.33
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19014058 0.90 EPHX2 (0.32) CCR2JAK2JAK1
SCHEMBL20682206 0.81 CCR2 (0.34) CCR2JAK2JAK1
SCHEMBL14211363 0.79 CCR2 (0.32) CCR2
SCHEMBL19013670 0.77 EPHX2 (0.34) CCR2
SCHEMBL19014535 0.74 CCR2 (0.43) CCR2JAK2JAK1
SCHEMBL19014504 0.73 JAK1 (0.37) CCR2JAK2JAK1
SCHEMBL19014086 0.73 NPC1 (0.34) CCR2JAK1
SCHEMBL19014405 0.73 NPC1 (0.32) CCR2
SCHEMBL20682199 0.71 ATM (0.33) CCR2JAK2JAK1
SCHEMBL19013820 0.71 JAK2 (0.39) CCR2JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017103188-A1 THERAPEUTIC COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-06-22 WO disclosed